SCHEMBL7980841

SCHEMBL7980841

CCOC(=O)[C@@H](N)Cc1cnc2ccccc2c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.50
CYP2C9 P11712 1/20 0.50
HIF1A Q16665 1/20 0.50
TPH1 P17752 3/20 0.47
MMP9 P14780 2/20 0.44
MMP1 P03956 1/20 0.44
FCER2 P06734 1/20 0.44
MMP3 P08254 1/20 0.44
KDM4E B2RXH2 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
ALDH1A1 P00352 1/20 0.43
LNPEP Q9UIQ6 1/20 0.43
ACACB O00763 1/20 0.42
KMT2A Q03164 2/20 0.42
PDE10A Q9Y233 1/20 0.42
MEN1 O00255 1/20 0.42
AKT1 P31749 2/20 0.42
NOTUM Q6P988 1/20 0.42
MMP2 P08253 1/20 0.41
MMP8 P22894 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8882758 0.99 CYP1A2 (0.49) CYP1A2CYP2C9HIF1ATPH1MMP9
Hydrochloric Acid SCHEMBL8882757 0.99 CYP1A2 (0.49) CYP1A2CYP2C9HIF1ATPH1MMP9
SCHEMBL8298247 0.88 TPH1 (0.50) CYP1A2TPH1MMP9MMP1FCER2
SCHEMBL9727511 0.88 TPH1 (0.50) CYP1A2TPH1MMP9MMP1FCER2
SCHEMBL15446279 0.85 CYP1A2 (0.48) CYP1A2CYP2C9HIF1AMMP9MMP1
SCHEMBL32662274 0.84 TPH1 (0.45) CYP1A2TPH1MMP9MMP1FCER2
SCHEMBL28978417 0.84 ACACB (0.47) FCER2KDM4ESMN1; SMN2ALDH1A1ACACB
SCHEMBL8884049 0.83 ALDH1A1 (0.53) CYP1A2TPH1KDM4ESMN1; SMN2ALDH1A1
Hydrochloric Acid SCHEMBL31407619 0.83 TPH1 (0.44) CYP1A2TPH1MMP9MMP1FCER2
SCHEMBL287073 0.82 TPH1 (0.62) HIF1ATPH1MMP9MMP1FCER2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6294549-B1 COMPOUNDS USEFUL FOR INHIBITING RESTENOSIS, ANGIOGENESIS, ATHEROSCLEROSIS, DIABETIC RETINOPATHY, MACULAR DEGENERATION, INFLAMMATION OR TUMOR GROWTH. MERCK & CO., INC. 2001-09-25 US disclosed
US-5639885-A Redox amino acids and peptides containing them UNIVERSITY OF FLORIDA (US) 1997-06-17 US disclosed
EP-0293071-B1 REDOX AMINO ACIDS AND PEPTIDES CONTAINING THEM UNIVERSITY OF FLORIDA (US) 1993-09-01 EP disclosed
US-5079366-A To derivatize pharmaceutical peptides for transport across the blood/brain barrier UNIVERSITY OF FLORIDA (US) 1992-01-07 US disclosed
US-4888427-A DIHYDROPYRIDINE-PYRIDINIUM SALT REDOX SYSTEM UNIVERSITY OF FLORIDA (US) 1989-12-19 US disclosed
EP-0293071-A1 Redox amino acids and peptides containing them UNIVERSITY OF FLORIDA (US) 1988-11-30 EP disclosed