SCHEMBL7981086

SCHEMBL7981086

CCOC(=O)Cc1cn2ccncc2n1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 10/20 0.44
ALDH1A1 P00352 9/20 0.44
POLB P06746 4/20 0.43
TDP1 Q9NUW8 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
HRH4 Q9H3N8 1/20 0.42
HPGD P15428 3/20 0.41
GAA P10253 2/20 0.41
CASP1 P29466 2/20 0.41
CASP7 P55210 2/20 0.41
HSD17B10 Q99714 2/20 0.41
ALOX15 P16050 1/20 0.41
MEN1 O00255 4/20 0.40
KMT2A Q03164 4/20 0.40
MAPT P10636 3/20 0.39
ESR1 P03372 1/20 0.39
RECQL P46063 1/20 0.39
ESR2 Q92731 1/20 0.39
DRD2 P14416 1/20 0.39
DRD4 P21917 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1668064 0.80 ALDH1A1 (0.60) KDM4EALDH1A1POLBTDP1L3MBTL1
SCHEMBL15230641 0.78 KDM4E (0.71) KDM4EALDH1A1POLBTDP1L3MBTL1
SCHEMBL2922016 0.78 KDM4E (0.63) KDM4EALDH1A1POLBL3MBTL1HRH4
SCHEMBL20533689 0.77 KDM4E (0.43) KDM4EALDH1A1POLBTDP1L3MBTL1
SCHEMBL20985955 0.76 KDM4E (0.53) KDM4EALDH1A1POLBTDP1L3MBTL1
SCHEMBL14912238 0.76 KDM4E (0.53) KDM4EALDH1A1POLBTDP1L3MBTL1
SCHEMBL15068790 0.76 KDM4E (0.49) KDM4EALDH1A1POLBTDP1L3MBTL1
SCHEMBL12223303 0.76 DRD2 (0.47) KDM4EALDH1A1POLBTDP1L3MBTL1
SCHEMBL16442152 0.75 KDM4E (0.52) KDM4EALDH1A1POLBTDP1L3MBTL1
SCHEMBL20595928 0.75 KDM4E (0.43) KDM4EALDH1A1POLBHPGDGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6174877-B1 EXCELLANT BACTERICIDES, ORAL ABSORBABILITY AND STABILITY; IMPROVE THE STABILITY TO RENAL DEHYDROPEPTIDASE I (DHP-I); 2-(2-(N-HETEROCYCLIC-ETHYLTHIO-) DERIVATIVES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-01-16 US disclosed
EP-0876370-A1 CARBAPENEM COMPOUNDS, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1998-11-11 EP disclosed
WO-1997025325-A1 CARBAPENEM COMPOUNDS, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-07-17 WO disclosed