SCHEMBL7982243

SCHEMBL7982243

O=C(Nc1oc(-c2ccccc2O)nc1-c1csc(-c2ccccc2)c1)c1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 6/20 0.48
FLT1 P17948 1/20 0.48
FLT4 P35916 1/20 0.48
ABCG2 Q9UNQ0 1/20 0.40
TYR P14679 1/20 0.40
RRM1 P23921 1/20 0.40
RRM2B Q7LG56 1/20 0.40
NPC1 O15118 3/20 0.39
RAB9A P51151 3/20 0.39
MAPT P10636 2/20 0.39
NPSR1 Q6W5P4 2/20 0.39
PTPN5 P54829 1/20 0.39
SMN1; SMN2 Q16637 3/20 0.39
GAA P10253 2/20 0.39
HSD17B10 Q99714 1/20 0.38
ALDH1A1 P00352 2/20 0.38
KDM4E B2RXH2 2/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
POLB P06746 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7744649 0.87 KDR (0.58) KDRFLT1FLT4ABCG2NPC1
SCHEMBL7746598 0.79 KDR (0.58) KDRFLT1FLT4ABCG2RRM1
SCHEMBL7746601 0.78 KDR (0.53) KDRFLT1FLT4ABCG2NPC1
SCHEMBL7744781 0.76 ADCY1 (0.47) KDRFLT1FLT4ABCG2TYR
SCHEMBL7744059 0.76 KDR (0.53) KDRFLT1FLT4NPC1RAB9A
SCHEMBL7746570 0.75 KDR (0.49) KDRFLT1FLT4ABCG2TYR
SCHEMBL7985537 0.75 KDR (0.53) KDRFLT1FLT4MAPTNPSR1
SCHEMBL4737638 0.75 KDR (0.55) KDRFLT1FLT4ABCG2NPC1
SCHEMBL7969519 0.74 KDR (0.44) KDRFLT1FLT4TYRRRM1
SCHEMBL7746649 0.74 KDR (0.47) KDRFLT1FLT4ABCG2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6228871-B1 THIAZOLE OR OXAZOLE DERIVATIVE TYROSINE KINASE INHIBITORS; ANTICARCINOGENIC AGENTS; AUTOIMMUNE DISEASES; DIABETIC RETINOPATHY MERCK & CO., INC. 2001-05-08 US claimed