SCHEMBL7982846

SCHEMBL7982846

CC(=O)Nc1oc(-c2ccc(-c3cccc(F)c3)cc2O)nc1C1=CC(=S)CC=C1

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KDR P35968 7/20 0.49
FLT1 P17948 1/20 0.46
FLT4 P35916 1/20 0.46
ADORA3 P0DMS8 2/20 0.38
ADORA2A P29274 2/20 0.38
ADORA2B P29275 2/20 0.38
ADORA1 P30542 2/20 0.38
TOP2A P11388 1/20 0.34
TRPM8 Q7Z2W7 4/20 0.32
ALOX15 P16050 1/20 0.32
GPR35 Q9HC97 1/20 0.32
NQO2 P16083 1/20 0.31
HSD17B1 P14061 1/20 0.31
HSD17B2 P37059 1/20 0.31
EGLN1 Q9GZT9 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7744769 0.91 KDR (0.53) KDRFLT1FLT4ADORA2AADORA1
SCHEMBL7986526 0.89 KDR (0.42) KDRFLT1FLT4ADORA3ADORA2A
SCHEMBL7982717 0.88 KDR (0.44) KDRFLT1FLT4ADORA3ALOX15
SCHEMBL7739072 0.87 KDR (0.43) KDRFLT1FLT4NQO2
SCHEMBL7981120 0.86 KDR (0.47) KDRFLT1FLT4ALOX15
SCHEMBL7980279 0.85 KDR (0.47) KDRFLT1FLT4ADORA3
SCHEMBL7986670 0.82 KDR (0.50) KDRFLT1FLT4ADORA3ADORA2A
SCHEMBL7746568 0.82 KDR (0.41) KDRFLT1FLT4
SCHEMBL7979682 0.80 KDR (0.46) KDRFLT1FLT4ALOX15
SCHEMBL7969457 0.79 KDR (0.42) KDRFLT1FLT4ADORA2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6228871-B1 THIAZOLE OR OXAZOLE DERIVATIVE TYROSINE KINASE INHIBITORS; ANTICARCINOGENIC AGENTS; AUTOIMMUNE DISEASES; DIABETIC RETINOPATHY MERCK & CO., INC. 2001-05-08 US claimed