SCHEMBL7969457

SCHEMBL7969457

O=C(Nc1oc(-c2ccc(-c3cccc(Cl)c3)cc2O)nc1C1=CC(=S)CC=C1)c1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 2/20 0.42
ADORA1 P30542 2/20 0.38
FLT1 P17948 1/20 0.38
FLT4 P35916 1/20 0.38
ADORA2A P29274 1/20 0.38
MAPT P10636 4/20 0.38
HSP90AA1 P07900 1/20 0.36
HSP90AB1 P08238 1/20 0.36
GRM5 P41594 1/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
SERPINE1 P05121 2/20 0.36
GAA P10253 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
KDM4E B2RXH2 1/20 0.34
LMNA P02545 1/20 0.34
CYP1A2 P05177 1/20 0.34
POLB P06746 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7746568 0.93 KDR (0.41) KDRFLT1FLT4MAPTGAA
SCHEMBL7986526 0.90 KDR (0.42) KDRADORA1FLT1FLT4ADORA2A
SCHEMBL7986013 0.89 KDR (0.39) KDRFLT1FLT4MAPTNPC1
SCHEMBL7739003 0.88 HPN (0.44) KDRFLT1FLT4MAPTRAB9A
SCHEMBL7969509 0.87 MCL1 (0.38) KDRFLT1FLT4MAPTNPC1
SCHEMBL7980106 0.86 KDR (0.42) KDRFLT1FLT4MAPTHSP90AA1
SCHEMBL7744769 0.84 KDR (0.53) KDRADORA1FLT1FLT4ADORA2A
SCHEMBL7744059 0.83 KDR (0.53) KDRADORA1FLT1FLT4ADORA2A
SCHEMBL7987348 0.82 KDR (0.44) KDRADORA1FLT1FLT4ADORA2A
SCHEMBL7982846 0.79 KDR (0.49) KDRADORA1FLT1FLT4ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6228871-B1 THIAZOLE OR OXAZOLE DERIVATIVE TYROSINE KINASE INHIBITORS; ANTICARCINOGENIC AGENTS; AUTOIMMUNE DISEASES; DIABETIC RETINOPATHY MERCK & CO., INC. 2001-05-08 US claimed