SCHEMBL7986526

SCHEMBL7986526

O=C(Nc1oc(-c2ccc(-c3cccc(F)c3)cc2O)nc1C1=CC(=S)CC=C1)c1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 2/20 0.42
FLT1 P17948 1/20 0.38
FLT4 P35916 1/20 0.38
ADCY1 Q08828 5/20 0.37
ADCY8 P40145 3/20 0.37
KMT2A Q03164 3/20 0.36
HPGD P15428 3/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
SMN1; SMN2 Q16637 4/20 0.34
GAA P10253 2/20 0.34
ADORA3 P0DMS8 1/20 0.34
ADORA2A P29274 1/20 0.34
ADORA2B P29275 1/20 0.34
ADORA1 P30542 1/20 0.34
MAPT P10636 2/20 0.34
MEN1 O00255 2/20 0.33
POLB P06746 2/20 0.33
TP53 P04637 2/20 0.33
KCNK3 O14649 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7746568 0.93 KDR (0.41) KDRFLT1FLT4ADCY1ADCY8
SCHEMBL7969457 0.90 KDR (0.42) KDRFLT1FLT4KMT2AHPGD
SCHEMBL7982846 0.89 KDR (0.49) KDRFLT1FLT4ADORA3ADORA2A
SCHEMBL7986013 0.89 KDR (0.39) KDRFLT1FLT4KMT2AHPGD
SCHEMBL7739003 0.88 HPN (0.44) KDRFLT1FLT4KMT2ARAB9A
SCHEMBL7969509 0.87 MCL1 (0.38) KDRFLT1FLT4KMT2AHPGD
SCHEMBL7980106 0.86 KDR (0.42) KDRFLT1FLT4KMT2AHPGD
SCHEMBL7744769 0.84 KDR (0.53) KDRFLT1FLT4NPC1RAB9A
SCHEMBL7744069 0.79 KDR (0.40) KDRFLT1FLT4HPGDNPC1
SCHEMBL7982717 0.77 KDR (0.44) KDRFLT1FLT4KMT2AHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6228871-B1 THIAZOLE OR OXAZOLE DERIVATIVE TYROSINE KINASE INHIBITORS; ANTICARCINOGENIC AGENTS; AUTOIMMUNE DISEASES; DIABETIC RETINOPATHY MERCK & CO., INC. 2001-05-08 US claimed