SCHEMBL7983253

SCHEMBL7983253

Cc1cccc(Cl)c1-c1ncc2c(N)nc3cc(NCc4cccs4)ccc3n12

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 10/20 0.52
NPC1 O15118 9/20 0.52
ALDH1A1 P00352 8/20 0.52
RAB9A P51151 8/20 0.52
SMN1; SMN2 Q16637 6/20 0.52
HTT P42858 2/20 0.52
MAPT P10636 7/20 0.49
HPGD P15428 5/20 0.49
CYP1A2 P05177 4/20 0.49
CYP3A4 P08684 4/20 0.49
CYP2D6 P10635 4/20 0.49
CYP2C19 P33261 4/20 0.49
CYP2C9 P11712 3/20 0.49
POLB P06746 2/20 0.49
GAA P10253 2/20 0.48
LMNA P02545 6/20 0.46
TDP1 Q9NUW8 4/20 0.46
TSHR P16473 5/20 0.42
ALOX15 P16050 2/20 0.42
L3MBTL1 Q9Y468 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7969620 0.91 KDM4E (0.42) KDM4ENPC1ALDH1A1RAB9ASMN1; SMN2
SCHEMBL7981780 0.85 NPC1 (0.43) KDM4ENPC1ALDH1A1RAB9ASMN1; SMN2
SCHEMBL7983693 0.85 LCK (0.43) NPC1RAB9AMAPTGAAEGFR
SCHEMBL7981250 0.82 PDE2A (0.40)
SCHEMBL7982709 0.81 LCK (0.53)
SCHEMBL7981128 0.80 LCK (0.54) KMT2A
SCHEMBL7982930 0.79 LCK (0.51) KMT2A
SCHEMBL7983879 0.79 FGFR1 (0.55) EGFR
SCHEMBL7983214 0.78 LCK (0.51) EGFRKMT2A
SCHEMBL7983712 0.78 PDE2A (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6235740-B1 AUTOIMMUNE DISEASES; ANTIPROLIFERATION AGENTS BRISTOL-MYERS SQUIBB CO. 2001-05-22 US claimed
US-6235740-B1 AUTOIMMUNE DISEASES; ANTIPROLIFERATION AGENTS BRISTOL-MYERS SQUIBB CO. 2001-05-22 US disclosed