SCHEMBL7981780

SCHEMBL7981780

Cc1cccc(Cl)c1-c1ncc2c(N)nc3cc(NCc4ccccc4)ccc3n12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 9/20 0.43
RAB9A P51151 9/20 0.43
DHFR P00374 2/20 0.40
KDM4E B2RXH2 5/20 0.40
ALDH1A1 P00352 5/20 0.40
MAPT P10636 4/20 0.40
PKM P14618 2/20 0.40
TDP1 Q9NUW8 2/20 0.40
GAA P10253 2/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
TP53 P04637 3/20 0.39
TSHR P16473 1/20 0.39
HTT P42858 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
FGFR1 P11362 1/20 0.39
GFER P55789 1/20 0.39
HSD17B10 Q99714 3/20 0.38
THRB P10828 1/20 0.38
PDE2A O00408 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7983693 0.88 LCK (0.43) NPC1RAB9ADHFRMAPTGAA
SCHEMBL7983253 0.85 KDM4E (0.52) NPC1RAB9AKDM4EALDH1A1MAPT
SCHEMBL7981250 0.85 PDE2A (0.40) FGFR1PDE2A
SCHEMBL7982709 0.84 LCK (0.53) FGFR1PDE2A
SCHEMBL7987014 0.83 LCK (0.45) FGFR1PDE2A
SCHEMBL7981128 0.83 LCK (0.54) KMT2AFGFR1
SCHEMBL7980082 0.82 ROCK2 (0.45) MAPTTP53SMN1; SMN2
SCHEMBL7982930 0.82 LCK (0.51) KMT2AFGFR1PDE2A
SCHEMBL7983214 0.81 LCK (0.51) KMT2AFGFR1
SCHEMBL7983712 0.81 PDE2A (0.39) FGFR1PDE2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6235740-B1 AUTOIMMUNE DISEASES; ANTIPROLIFERATION AGENTS BRISTOL-MYERS SQUIBB CO. 2001-05-22 US claimed
US-6235740-B1 AUTOIMMUNE DISEASES; ANTIPROLIFERATION AGENTS BRISTOL-MYERS SQUIBB CO. 2001-05-22 US disclosed