SCHEMBL7983354

SCHEMBL7983354

O=C(O)C1=Cc2cnc3cccc(n23)S1

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7972990 0.98
SCHEMBL13763779 0.81 APOBEC3A (0.40)
SCHEMBL7983803 0.79 HCAR2 (0.35)
SCHEMBL7985758 0.73 NPC1 (0.42)
Hydrochloric Acid SCHEMBL7972479 0.72 NPC1 (0.41)
SCHEMBL8527068 0.71 L3MBTL1 (0.48)
Hydrochloric Acid SCHEMBL7971798 0.71 CHRM1 (0.40)
SCHEMBL7986609 0.70 DRD3 (0.44)
Hydrochloric Acid SCHEMBL7983228 0.70 HDAC3 (0.50)
Hydrochloric Acid SCHEMBL7982276 0.69 GAA (0.44)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-10226687-A None JP disclosed
JP-11005795-A None JP disclosed
US-6235731-B1 REDUCING BLOOD LIPIDS, SUGARS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-05-22 US disclosed
EP-0915888-A1 FUSED IMIDAZOPYRIDINE DERIVATIVES AS ANTIHYPERLIPIDEMIC AGENTS Takeda Chemical Industries, Ltd. (JP) 1999-05-19 EP disclosed
JP-H115795-A PRODUCTION OF PIPERIDINE DERIVATIVE TAKEDA CHEM IND LTD 1999-01-12 JP disclosed
JP-H10226687-A IMIDAZOPYRIDINE DERIVATIVE AND ITS PRODUCTION TAKEDA CHEM IND LTD 1998-08-25 JP disclosed
WO-1997040051-A1 FUSED IMIDAZOPYRIDINE DERIVATIVES AS ANTIHYPERLIPIDEMIC AGENTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-10-30 WO disclosed