SCHEMBL7983383

SCHEMBL7983383

COc1cc(CN2CCC(CCO)(Cc3cccc(F)c3)C2=O)cc(OC)c1OC

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.42
TP53 P04637 1/20 0.41
GAA P10253 1/20 0.41
ALDH1A1 P00352 2/20 0.39
MAPK1 P28482 1/20 0.39
KDM4E B2RXH2 1/20 0.39
HTT P42858 1/20 0.39
HRH1 P35367 1/20 0.38
ACHE P22303 1/20 0.37
MEN1 O00255 1/20 0.37
USP2 O75604 1/20 0.37
LMNA P02545 1/20 0.37
THRB P10828 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C9 P11712 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6992507 0.89 ALDH1A1 (0.45) TP53ALDH1A1MAPK1KDM4EHTT
SCHEMBL6999204 0.89 MAPK1 (0.46) KMT2AGAAALDH1A1MAPK1ACHE
SCHEMBL7956133 0.87 KDM4E (0.43) KMT2AALDH1A1MAPK1KDM4EHTT
SCHEMBL7981028 0.87 TP53 (0.39) KMT2ATP53GAAALDH1A1MAPK1
SCHEMBL7961053 0.86 MEN1 (0.42) KMT2AALDH1A1MAPK1KDM4EHTT
SCHEMBL7971732 0.84 HRH1 (0.38) KMT2ATP53GAAALDH1A1MAPK1
SCHEMBL6998261 0.84 SMN1; SMN2 (0.46) KMT2AGAAALDH1A1MAPK1HTT
SCHEMBL7954561 0.84 MEN1 (0.40) KMT2AGAAMAPK1MEN1USP2
SCHEMBL7495346 0.84 ALDH1A1 (0.43) TP53ALDH1A1MAPK1KDM4EHTT
SCHEMBL6995389 0.83 KMT2A (0.39) KMT2AMAPK1HTTMEN1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6211199-B1 HISTAMINE AND TACHYKININ RECEPTOR ANTAGONISTS; ANTIASTHMATICS, ANTIEMETICS; RESPIRATORY SYSTEM DISORDERS, INFLAMMATORY BOWEL DISEASE, CONJUNCTIVITIS AVENTIS PHARMACEUTICALS INC. 2001-04-03 US disclosed