SCHEMBL7981028

SCHEMBL7981028

COc1cc(CN2CCC(CCOS(C)(=O)=O)(Cc3cccc(F)c3)C2=O)cc(OC)c1OC

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.39
GAA P10253 1/20 0.39
ALDH1A1 P00352 2/20 0.38
KDM4E B2RXH2 1/20 0.38
HTT P42858 1/20 0.38
KMT2A Q03164 2/20 0.38
HRH1 P35367 1/20 0.36
MEN1 O00255 1/20 0.35
ACHE P22303 1/20 0.35
MAPK1 P28482 1/20 0.35
POLB P06746 1/20 0.35
USP2 O75604 1/20 0.34
LMNA P02545 1/20 0.34
THRB P10828 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6996096 0.90 ALDH1A1 (0.44) TP53ALDH1A1KDM4EHTTHRH1
SCHEMBL6998268 0.90 MAPK1 (0.41) GAAALDH1A1KDM4EHTTKMT2A
SCHEMBL7983383 0.87 KMT2A (0.42) TP53GAAALDH1A1KDM4EHTT
SCHEMBL6992505 0.86 L3MBTL1 (0.43) GAAALDH1A1HTTKMT2AMEN1
SCHEMBL6997482 0.85 ALDH1A1 (0.42) TP53ALDH1A1KDM4EHTTHRH1
SCHEMBL6994509 0.84 KMT2A (0.37) GAAALDH1A1KDM4EHTTKMT2A
SCHEMBL7971732 0.84 HRH1 (0.38) TP53GAAALDH1A1KDM4EHTT
SCHEMBL27404103 0.84 MAPK1 (0.40) GAAALDH1A1KDM4EHTTKMT2A
SCHEMBL6997994 0.83 CYP2D6 (0.37) ALDH1A1KDM4EHTTKMT2AMEN1
Fluorobenzene SCHEMBL27405662 0.81 HTT (0.44) GAAALDH1A1KDM4EHTTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6211199-B1 HISTAMINE AND TACHYKININ RECEPTOR ANTAGONISTS; ANTIASTHMATICS, ANTIEMETICS; RESPIRATORY SYSTEM DISORDERS, INFLAMMATORY BOWEL DISEASE, CONJUNCTIVITIS AVENTIS PHARMACEUTICALS INC. 2001-04-03 US disclosed