SCHEMBL7983633

SCHEMBL7983633

CCCC(N)C(=S)c1cc(C(=O)OC)sc1SC

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.34
PKM P14618 1/20 0.34
HPGD P15428 4/20 0.33
MAPK1 P28482 2/20 0.33
TSHR P16473 1/20 0.33
ATM Q13315 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
ALDH1A1 P00352 3/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2C19 P33261 1/20 0.32
ERAP2 Q6P179 2/20 0.32
LNPEP Q9UIQ6 2/20 0.32
KEAP1 Q14145 1/20 0.32
NFE2L2 Q16236 1/20 0.32
C1S P09871 1/20 0.31
S100A4 P26447 1/20 0.31
KDM4E B2RXH2 2/20 0.30
LMNA P02545 1/20 0.30
MAPT P10636 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6921023 0.78 CSNK2A2 (0.38) HPGDMAPK1TSHRATMNPSR1
SCHEMBL7983624 0.75 HPGD (0.34) POLBPKMHPGDMAPK1TSHR
SCHEMBL6925163 0.73 KEAP1 (0.47) POLBPKMHPGDMAPK1TSHR
SCHEMBL6925132 0.71 KEAP1 (0.37) PKMHPGDMAPK1TSHRATM
SCHEMBL6920646 0.70 ALDH1A1 (0.40) HPGDMAPK1ALDH1A1KEAP1NFE2L2
SCHEMBL5839757 0.69 KEAP1 (0.41) HPGDMAPK1TSHRATMNPSR1
SCHEMBL7983629 0.68 CSNK2A2 (0.31) KEAP1NFE2L2C1S
SCHEMBL6925185 0.67 KDM4E (0.48) HPGDMAPK1TSHRATMNPSR1
SCHEMBL6923952 0.66 KEAP1 (0.41) PKMHPGDMAPK1TSHRATM
SCHEMBL7983631 0.66 ALDH1A1 (0.33) HPGDMAPK1TSHRATMNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6291514-B1 Heteroaryl amidines, methylamidines and guanidines, preparation thereof, and use thereof as protease inhibitors 3-DIMENSIONAL PHARMACEUTICALS, INC. 2001-09-18 US disclosed