SCHEMBL7984023

SCHEMBL7984023

COc1cc(COC23CC4CC(CC(C4)C2)C3)nn1C1CCCCC1.Oc1cc(COC23CC4CC(CC(C4)C2)C3)nn1C1CCCCC1

nearest known ligand 0.36

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 1/20 0.36
SIGMAR1 Q99720 1/20 0.32
SCN9A Q15858 1/20 0.31
ALDH1A1 P00352 1/20 0.31
CNR2 P34972 1/20 0.31
CCKBR P32239 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6497641 0.94 PTGS2 (0.39) PTGS2SIGMAR1SCN9ACNR2CCKBR
SCHEMBL6490137 0.91 PTGS2 (0.38) PTGS2SIGMAR1SCN9AALDH1A1CNR2
SCHEMBL6500868 0.82 PTGS2 (0.33) PTGS2SCN9A
SCHEMBL6489101 0.68 CNR2 (0.31) CNR2
SCHEMBL30088717 0.67 SIGMAR1 (0.36) PTGS2SIGMAR1ALDH1A1
SCHEMBL6487195 0.65 SLC16A3 (0.38) ALDH1A1CNR2
SCHEMBL6064596 0.65 ALDH1A1 (0.37) SCN9AALDH1A1CNR2CCKBR
SCHEMBL6065524 0.64 CNR2 (0.37) SCN9AALDH1A1CNR2CCKBR
SCHEMBL11451345 0.64 RET (0.34) PTGS2SIGMAR1ALDH1A1
SCHEMBL7984267 0.63 CNR2 (0.36) SIGMAR1CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001090078-A1 PYRAZOLE DERIVATIVES AND THEIR USE AS GASTRIN AND CHOLECYSTOKIN IN RECEPTOR LIGANDS JAMES BLACK FOUNDATION LIMITED (GB) 2001-11-29 WO disclosed