SCHEMBL7984142

SCHEMBL7984142

Cc1cc(C#Cc2ccc(O)c(CC(=O)O)c2)ccc1C1(OCc2ccccc2)CC1

nearest known ligand 0.35

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 1/20 0.35
FFAR1 O14842 7/20 0.34
CYP26A1 O43174 1/20 0.34
CYP3A4 P08684 1/20 0.34
RARA P10276 1/20 0.34
RARB P10826 1/20 0.34
RARG P13631 1/20 0.34
CRABP2 P29373 1/20 0.34
PTGER1 P34995 1/20 0.33
PTGER4 P35408 1/20 0.33
PTGER3 P43115 1/20 0.33
PTGER2 P43116 1/20 0.33
EGFR P00533 1/20 0.33
FFAR4 Q5NUL3 2/20 0.33
LMNA P02545 1/20 0.33
HNF4A P41235 1/20 0.33
RXRA P19793 1/20 0.32
RXRB P28702 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5736361 0.88 FFAR1 (0.49) AKR1B1FFAR1CYP26A1CYP3A4RARA
SCHEMBL7980612 0.83 MCL1 (0.37) CYP26A1CYP3A4RARARARBRARG
SCHEMBL5736240 0.82 RARB (0.53) CYP26A1CYP3A4RARARARBRARG
SCHEMBL5737152 0.81 FFAR1 (0.48) AKR1B1FFAR1CYP26A1CYP3A4RARA
SCHEMBL5736923 0.79 SMN1; SMN2 (0.46) CYP26A1CYP3A4RARARARBRARG
SCHEMBL6425926 0.79 ACACB (0.42) FFAR1CYP26A1CYP3A4RARARARB
SCHEMBL5736510 0.76 OPRM1 (0.33)
SCHEMBL5736289 0.76 OPRM1 (0.35)
SCHEMBL5735372 0.75 RARB (0.52) CYP26A1CYP3A4RARARARBRARG
SCHEMBL7970709 0.75 RARB (0.39) FFAR1CYP26A1CYP3A4RARARARB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6303785-B1 SUBSTITUTED N-CYCLOPROPYLTETRAHYDROISOQUINOLINES ALLERGAN SALES, INC. 2001-10-16 US disclosed