SCHEMBL6425926

SCHEMBL6425926

Cc1cc(C#Cc2ccc(C(C)C(=O)O)cc2)ccc1C1(OCc2ccccc2)CC1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACACB O00763 5/20 0.42
AKR1C3 P42330 3/20 0.37
AKR1C2 P52895 2/20 0.37
FFAR1 O14842 2/20 0.37
PTGS2 P35354 5/20 0.37
RARB P10826 2/20 0.37
CYP26A1 O43174 1/20 0.37
CYP3A4 P08684 1/20 0.37
RARA P10276 1/20 0.37
RARG P13631 1/20 0.37
CRABP2 P29373 1/20 0.37
PTGES O14684 2/20 0.35
PTGS1 P23219 3/20 0.34
LMNA P02545 2/20 0.34
CYP2C9 P11712 2/20 0.34
CXCR1 P25024 2/20 0.34
CXCR2 P25025 2/20 0.34
ALOX5 P09917 2/20 0.34
ALB P02768 1/20 0.34
ESR1 P03372 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6425907 0.89 ACACB (0.41) ACACBAKR1C3AKR1C2FFAR1PTGS2
SCHEMBL5736240 0.85 RARB (0.53) RARBCYP26A1CYP3A4RARARARG
SCHEMBL6427660 0.85 OPRM1 (0.44) ACACBAKR1C3AKR1C2FFAR1PTGS2
SCHEMBL6426294 0.84 RARB (0.37) ACACBAKR1C3AKR1C2FFAR1PTGS2
SCHEMBL5736361 0.84 FFAR1 (0.49) FFAR1RARBCYP26A1CYP3A4RARA
SCHEMBL6426262 0.83 RARB (0.38) ACACBAKR1C3AKR1C2FFAR1PTGS2
SCHEMBL5736923 0.82 SMN1; SMN2 (0.46) ACACBRARBCYP26A1CYP3A4RARA
SCHEMBL7980612 0.80 MCL1 (0.37) RARBCYP26A1CYP3A4RARARARG
SCHEMBL7984142 0.79 AKR1B1 (0.35) FFAR1RARBCYP26A1CYP3A4RARA
SCHEMBL6426280 0.78 PTGS2 (0.41) ACACBAKR1C3AKR1C2PTGS2RARB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6855512-B2 Methods for identifying inhibitors of cytochrome P450RAI ALLERGAN, INC. (US) 2005-02-15 US disclosed
US-6369261-B1 CYCLOPROPYLBENZENE DERIVATIVE OF ACIDS OR ESTERS ALLERGAN SALES, INC. 2002-04-09 US disclosed
US-6369225-B1 ENZYME INHIBITORS ALLERGAN SALES, INC. 2002-04-09 US disclosed
US-6303785-B1 SUBSTITUTED N-CYCLOPROPYLTETRAHYDROISOQUINOLINES ALLERGAN SALES, INC. 2001-10-16 US disclosed