SCHEMBL7984550

SCHEMBL7984550

COc1ccc2c(c1)N(C(=O)O)CC2

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 2/20 0.60
BIRC2 Q13490 1/20 0.55
RAB9A P51151 6/20 0.52
SMN1; SMN2 Q16637 6/20 0.52
NPC1 O15118 4/20 0.50
MAPT P10636 3/20 0.50
PKM P14618 1/20 0.50
NFKB1 P19838 1/20 0.50
MAOB P27338 1/20 0.50
NFKB2 Q00653 1/20 0.50
RELA Q04206 1/20 0.50
HSD17B10 Q99714 1/20 0.49
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
DRD2 P14416 1/20 0.47
DRD1 P21728 1/20 0.47
DRD5 P21918 1/20 0.47
DRD3 P35462 1/20 0.47
MAPK1 P28482 1/20 0.47
ESR1 P03372 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30804503 0.91 HSD17B10 (0.60) NOTUMBIRC2RAB9ASMN1; SMN2NPC1
SCHEMBL2208006 0.88 NOTUM (0.78) NOTUMBIRC2RAB9ASMN1; SMN2NPC1
SCHEMBL26691241 0.86 NOTUM (0.58) NOTUMBIRC2RAB9ASMN1; SMN2NPC1
SCHEMBL17311751 0.85 LMNA (0.50) NOTUMBIRC2RAB9ASMN1; SMN2MEN1
SCHEMBL27165463 0.82 BIRC2 (0.60) NOTUMBIRC2RAB9ASMN1; SMN2NPC1
SCHEMBL26922623 0.82 SMN1; SMN2 (0.47) NOTUMBIRC2RAB9ASMN1; SMN2NPC1
SCHEMBL14230676 0.81 DRD2 (0.55) NOTUMBIRC2RAB9ASMN1; SMN2NPC1
SCHEMBL6960928 0.81 BIRC2 (0.58) NOTUMBIRC2RAB9ASMN1; SMN2NPC1
SCHEMBL6962584 0.80 BIRC2 (0.57) NOTUMBIRC2RAB9ASMN1; SMN2NPC1
SCHEMBL27165447 0.80 BIRC2 (0.57) NOTUMBIRC2RAB9ASMN1; SMN2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6274594-B1 ANTICONVULSANTS, ANALGESICS; NERUOPATHIC, CANCER AND DENTAL PAIN; SMITHKLINE BEECHAM P.L.C. (GB) 2001-08-14 US claimed
EP-1032570-A1 ISOQUINOLINE DERIVATIVES AND THEIR THERAPEUTICAL USE SMITHKLINE BEECHAM PLC (GB) 2000-09-06 EP claimed
WO-1999025709-A1 ISOQUINOLINE DERIVATIVES AND THEIR THERAPEUTICAL USE SMITHKLINE BEECHAM P.L.C. (GB) 1999-05-27 WO claimed
US-6274594-B1 ANTICONVULSANTS, ANALGESICS; NERUOPATHIC, CANCER AND DENTAL PAIN; SMITHKLINE BEECHAM P.L.C. (GB) 2001-08-14 US disclosed
EP-1032570-A1 ISOQUINOLINE DERIVATIVES AND THEIR THERAPEUTICAL USE SMITHKLINE BEECHAM PLC (GB) 2000-09-06 EP disclosed
WO-1999025709-A1 ISOQUINOLINE DERIVATIVES AND THEIR THERAPEUTICAL USE SMITHKLINE BEECHAM P.L.C. (GB) 1999-05-27 WO disclosed