SCHEMBL7984853

SCHEMBL7984853

Cc1c(Cn2cncc2C(=O)O)cccc1OCCNC(=O)OC(C)(C)C

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 1/20 0.46
CA12 O43570 2/20 0.38
CA1 P00915 2/20 0.38
CA2 P00918 2/20 0.38
CA9 Q16790 2/20 0.38
IDO1 P14902 1/20 0.37
BUB1 O43683 1/20 0.37
ADRB2 P07550 1/20 0.37
HTR1A P08908 1/20 0.37
BRD4 O60885 1/20 0.36
NQO2 P16083 1/20 0.36
CKS1B P61024 1/20 0.36
SKP1 P63208 1/20 0.36
SKP2 Q13309 1/20 0.36
DRD2 P14416 2/20 0.35
FNTA P49354 1/20 0.35
FNTB P49356 1/20 0.35
PGGT1B P53609 1/20 0.35
KCNH2 Q12809 1/20 0.35
EGFR P00533 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7995719 0.92 SCN9A (0.45) SCN9ACA12CA1CA2CA9
SCHEMBL7983762 0.81 SCN9A (0.44) SCN9ACA12CA1CA2CA9
SCHEMBL8001577 0.81 BRD4 (0.47) SCN9AADRB2BRD4
SCHEMBL7995803 0.80 SCN9A (0.44) SCN9ACA12CA1CA2CA9
SCHEMBL7994019 0.78 SCN9A (0.48) SCN9ACA12CA1CA2CA9
SCHEMBL7984848 0.78 SCN9A (0.43) SCN9ACA12CA1CA2CA9
SCHEMBL7995494 0.77 SCN9A (0.48) SCN9ACA12CA1CA2CA9
SCHEMBL7995700 0.77 SCN9A (0.43) SCN9ACA12CA1CA2CA9
SCHEMBL7983883 0.76 SCN9A (0.43) SCN9ACA12CA1CA2CA9
SCHEMBL20630423 0.74 SCN9A (0.51) SCN9ACA12CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001034578-A1 COMPOUNDS WITH ANTI-HELICOBACTER PYLORI ACTIVITY ASTRAZENECA AB (SE) 2001-05-17 WO claimed
WO-2001034578-A1 COMPOUNDS WITH ANTI-HELICOBACTER PYLORI ACTIVITY ASTRAZENECA AB (SE) 2001-05-17 WO disclosed