SCHEMBL7983883

SCHEMBL7983883

CNC(=O)c1cn(Cc2cccc(OCCNC(=O)OC(C)(C)C)c2C)cn1

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 1/20 0.43
CA12 O43570 2/20 0.37
CA1 P00915 2/20 0.37
CA2 P00918 2/20 0.37
CA9 Q16790 2/20 0.37
ADRB2 P07550 1/20 0.36
HTR1A P08908 1/20 0.36
NQO2 P16083 1/20 0.35
SUCNR1 Q9BXA5 1/20 0.34
IDO1 P14902 1/20 0.34
DRD2 P14416 1/20 0.34
BRD4 O60885 2/20 0.34
PDK2 Q15119 1/20 0.34
BUB1 O43683 1/20 0.34
KLKB1 P03952 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7983762 0.91 SCN9A (0.44) SCN9ACA12CA1CA2CA9
SCHEMBL7995700 0.90 SCN9A (0.43) SCN9ACA12CA1CA2CA9
SCHEMBL7983840 0.89 KLKB1 (0.38) KLKB1
SCHEMBL7997642 0.83 MAPT (0.42) KLKB1
SCHEMBL7998248 0.83 KLKB1 (0.35) HTR1ADRD2KLKB1
SCHEMBL7994180 0.83 KLKB1 (0.39) HTR1ADRD2KLKB1
SCHEMBL8001577 0.81 BRD4 (0.47) SCN9AADRB2BRD4
SCHEMBL7994019 0.77 SCN9A (0.48) SCN9ACA12CA1CA2CA9
SCHEMBL7984853 0.76 SCN9A (0.46) SCN9ACA12CA1CA2CA9
SCHEMBL7995494 0.76 SCN9A (0.48) SCN9ACA12CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001034578-A1 COMPOUNDS WITH ANTI-HELICOBACTER PYLORI ACTIVITY ASTRAZENECA AB (SE) 2001-05-17 WO disclosed