SCHEMBL7984894

SCHEMBL7984894

NC(=O)c1ccc(O)nc1N1CCNCC1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 2/20 0.40
ACVR1 Q04771 4/20 0.40
KDM4E B2RXH2 1/20 0.39
SYK P43405 2/20 0.38
TGFBR1 P36897 1/20 0.38
CHRNB2 P17787 1/20 0.38
CHRNA4 P43681 1/20 0.38
HRH4 Q9H3N8 1/20 0.38
ADRB2 P07550 1/20 0.38
NCF1 P14598 1/20 0.38
PLD1 Q13393 1/20 0.38
SRC P12931 1/20 0.37
HTR2C P28335 1/20 0.37
PRKD3 O94806 1/20 0.37
PRKD1 Q15139 1/20 0.37
PRKD2 Q9BZL6 1/20 0.37
HTR3E A5X5Y0 1/20 0.36
HTR3B O95264 1/20 0.36
ALDH1A1 P00352 1/20 0.36
HTR3A P46098 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7242650 0.84 NPC1 (0.49) PARP1KDM4EALDH1A1
SCHEMBL3453077 0.80 ADRB1 (0.48) PARP1ACVR1ADRB2HTR2CALDH1A1
SCHEMBL30945091 0.76 EPHX2 (0.52) KDM4EPLD1HTR2CALDH1A1PRKCA
SCHEMBL4538970 0.76 EPHX2 (0.52) KDM4EPLD1HTR2CALDH1A1PRKCA
Hydrochloric Acid SCHEMBL5901187 0.75 EPHX2 (0.51) KDM4EPLD1HTR2CALDH1A1PRKCA
SCHEMBL6651476 0.74 PIM1 (0.42) PARP1ACVR1TGFBR1PRKD3PRKD1
SCHEMBL2351827 0.72 CHRNB2 (0.41) PARP1ACVR1CHRNB2CHRNA4HRH4
SCHEMBL30572289 0.72 IKBKB (0.45) ACVR1KDM4ETGFBR1HTR2CPRKD3
SCHEMBL16613201 0.72 ADRB2 (0.52) PARP1KDM4EADRB2HTR2CPRKD3
SCHEMBL20998571 0.70 NPC1 (0.46) KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001077078-A1 NOVEL PYRIDONES AND THEIR USE AS MODULATORS OF SERINE HYDROLASE ENZYMES DALHOUSIE UNIVERSITY (CA) 2001-10-18 WO disclosed