SCHEMBL7985192

SCHEMBL7985192

O=[N+]([O-])c1ccc(N2CCCN(Cc3ccccc3)CC2)c(Cl)c1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.62
LMNA P02545 4/20 0.62
CYP2C19 P33261 2/20 0.61
CYP3A4 P08684 1/20 0.61
CYP2C9 P11712 1/20 0.61
HPGD P15428 1/20 0.59
MAPT P10636 7/20 0.56
CYP1A2 P05177 1/20 0.56
CYP2D6 P10635 1/20 0.56
TDP1 Q9NUW8 1/20 0.56
SMN1; SMN2 Q16637 3/20 0.56
MAPK1 P28482 2/20 0.56
NPBWR1 P48145 1/20 0.55
MCHR1 Q99705 1/20 0.55
L3MBTL1 Q9Y468 1/20 0.55
CASP1 P29466 1/20 0.54
CASP4 P49662 1/20 0.54
CASP5 P51878 1/20 0.54
CCR2 P41597 1/20 0.54
ACHE P22303 2/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3201205 0.88 ALDH1A1 (0.60) ALDH1A1LMNACYP2C19CYP3A4CYP2C9
SCHEMBL6449799 0.83 ALDH1A1 (0.64) ALDH1A1LMNACYP2C19CYP3A4CYP2C9
SCHEMBL5206645 0.83 POLB (0.68) ALDH1A1LMNAMAPTTDP1SMN1; SMN2
SCHEMBL6315934 0.81 ALDH1A1 (0.62) ALDH1A1LMNACYP2C19CYP3A4CYP2C9
SCHEMBL5393900 0.81 LMNA (0.67) ALDH1A1LMNACYP2C19CYP3A4CYP2C9
SCHEMBL6858096 0.81 MEN1 (0.65) ALDH1A1LMNACYP2C19CYP3A4CYP2C9
SCHEMBL6815260 0.80 GAA (0.69) ALDH1A1LMNACYP2C19CYP3A4CYP2C9
SCHEMBL19212110 0.80 ALDH1A1 (0.61) ALDH1A1LMNACYP2C19CYP3A4CYP2C9
SCHEMBL3957309 0.80 ALDH1A1 (0.70) ALDH1A1LMNACYP2C19CYP3A4CYP2C9
SCHEMBL11551872 0.80 KDM4E (0.57) ALDH1A1LMNAMAPTTDP1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6333320-B1 USEFUL AS DRUGS, ESPECIALLY AS AN ACTIVATED BLOOD COAGULATION FACTOR X INHIBITOR Yamanouchi Pharmaceutical Co. (JP) 2001-12-25 US disclosed
EP-1000936-A1 NOVEL HEXAHYDRO-1,4-DIAZEPINE DERIVATIVES OR SALTS THEREOF YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 2000-05-17 EP disclosed