Pirenzepine

Pirenzepine

SCHEMBL7985618

C=C.CN1CCN(CC(=O)N2c3ccccc3C(=O)Nc3cccnc32)CC1.Cl.Cl

nearest known ligand 0.98

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

CHRM1

The experimentally established mechanism targets of Pirenzepine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CHRM1 known ✓ P11229 2/20 0.96
LMNA P02545 2/20 0.98
GMNN O75496 1/20 0.98
APEX1 P27695 1/20 0.98
CHRM2 P08172 2/20 0.96
USP2 O75604 1/20 0.96
ALDH1A1 P00352 1/20 0.96
CYP1A2 P05177 1/20 0.96
CHRM4 P08173 1/20 0.96
CHRM5 P08912 1/20 0.96
CYP2D6 P10635 1/20 0.96
CHRM3 P20309 1/20 0.96

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Pirenzepine SCHEMBL30548470 0.99 LMNA (1.00) LMNAGMNNAPEX1CHRM2CHRM1
Pirenzepine SCHEMBL41704 0.99 LMNA (1.00) LMNAGMNNAPEX1CHRM2CHRM1
Pirenzepine SCHEMBL1462692 0.99 LMNA (1.00) LMNAGMNNAPEX1CHRM2CHRM1
Pirenzepine SCHEMBL5987941 0.98 LMNA (0.98) LMNAGMNNAPEX1CHRM2CHRM1
Pirenzepine SCHEMBL11415337 0.98 LMNA (0.98) LMNAGMNNAPEX1CHRM2CHRM1
Pirenzepine SCHEMBL9254860 0.98 LMNA (1.00) LMNAGMNNAPEX1CHRM2CHRM1
Pirenzepine SCHEMBL29793172 0.98 LMNA (1.00) LMNAGMNNAPEX1CHRM2CHRM1
Pirenzepine SCHEMBL41705 0.98 LMNA (1.00) LMNAGMNNAPEX1CHRM2CHRM1
Pirenzepine SCHEMBL30553045 0.98 LMNA (1.00) LMNAGMNNAPEX1CHRM2CHRM1
Pirenzepine SCHEMBL15300969 0.97 LMNA (0.98) LMNAGMNNAPEX1CHRM2CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000009316-A1 FIBEROPTIC CONDUIT AND PROCESSES OF MANUFACTURE LUMENYTE INTERNATIONAL CORPORATION (US) 2000-02-24 WO disclosed