SCHEMBL7985647

SCHEMBL7985647

CC(=O)N(c1ccccc1)c1ncccc1C

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.50
TSHR P16473 3/20 0.48
KMT2A Q03164 2/20 0.48
MEN1 O00255 1/20 0.48
GAA P10253 1/20 0.45
HDAC6 Q9UBN7 2/20 0.41
NPC1 O15118 3/20 0.41
RAB9A P51151 2/20 0.41
NPSR1 Q6W5P4 1/20 0.41
HTT P42858 1/20 0.41
ATM Q13315 1/20 0.41
APAF1 O14727 1/20 0.40
NOTUM Q6P988 1/20 0.40
NOS3 P29474 1/20 0.39
NOS1 P29475 1/20 0.39
NOS2 P35228 1/20 0.39
KDM4E B2RXH2 1/20 0.38
LMNA P02545 1/20 0.38
NAPRT Q6XQN6 1/20 0.38
P4HTM Q9NXG6 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7978954 0.86 ALDH1A1 (0.43) ALDH1A1TSHRKMT2AMEN1NPC1
SCHEMBL7985661 0.84 TSHR (0.43) ALDH1A1TSHRKMT2AMEN1GAA
SCHEMBL7985664 0.83 HDAC6 (0.44) ALDH1A1TSHRKMT2AGAAHDAC6
SCHEMBL7978926 0.83 ALDH1A1 (0.43) ALDH1A1TSHRKMT2AMEN1NPC1
SCHEMBL7978886 0.80 KMT2A (0.48) ALDH1A1TSHRKMT2AMEN1GAA
SCHEMBL8691853 0.79 KMT2A (0.41) ALDH1A1TSHRKMT2AMEN1GAA
SCHEMBL7978951 0.79 POLQ (0.42) ALDH1A1TSHRKMT2AMEN1GAA
Hydrochloric Acid SCHEMBL7846316 0.78 GAA (0.39) ALDH1A1TSHRKMT2AMEN1GAA
SCHEMBL7982076 0.78 ALDH1A1 (0.51) ALDH1A1TSHRKMT2AMEN1GAA
SCHEMBL15206612 0.78 TDP1 (0.51) ALDH1A1TSHRKMT2AMEN1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6235730-B1 ANTICHOLESTEROL AGENT, ANTILIPEMIC AGENT JAPAN TOBACCO, INC. (JP) 2001-05-22 US disclosed
CN-1252068-A 3-piperidyl-4-oxoquinazoline derivatives and pharmaceutical compositions containing the same JAPAN TOBACCO INC (JP) 2000-05-03 CN disclosed
EP-0970954-A1 3-PIPERIDYL-4-OXOQUINAZOLINE DERIVATIVES AND MEDICINCAL COMPOSITIONS CONTAINING THE SAME JAPAN TOBACCO INC. (JP) 2000-01-12 EP disclosed