SCHEMBL7978951

SCHEMBL7978951

CC(=O)N(c1ccccc1)c1ncccc1C(F)(F)F

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLQ O75417 2/20 0.42
ALDH1A1 P00352 3/20 0.40
OPRM1 P35372 1/20 0.40
SIGMAR1 Q99720 1/20 0.40
TRPV1 Q8NER1 1/20 0.40
HSD11B1 P28845 1/20 0.40
DHODH Q02127 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
KMO O15229 1/20 0.38
CTNNB1 P35222 1/20 0.38
WNT3A P56704 1/20 0.38
TSHR P16473 2/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
NFE2L2 Q16236 1/20 0.38
NPSR1 Q6W5P4 1/20 0.37
NPC1 O15118 2/20 0.37
APAF1 O14727 1/20 0.37
GAA P10253 1/20 0.36
CYP1A2 P05177 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7978954 0.81 ALDH1A1 (0.43) ALDH1A1OPRM1SIGMAR1TSHRMEN1
SCHEMBL7985647 0.79 ALDH1A1 (0.50) ALDH1A1HDAC6TSHRMEN1KMT2A
SCHEMBL7978926 0.78 ALDH1A1 (0.43) ALDH1A1TSHRMEN1KMT2ANPSR1
SCHEMBL2583273 0.77 POLQ (0.47) POLQALDH1A1TSHRMEN1KMT2A
SCHEMBL5242161 0.77 P2RY1 (0.39) ALDH1A1TSHRMEN1KMT2ANPSR1
SCHEMBL7978886 0.75 KMT2A (0.48) ALDH1A1TSHRMEN1KMT2ANPSR1
SCHEMBL8691853 0.74 KMT2A (0.41) ALDH1A1DHODHTSHRMEN1KMT2A
SCHEMBL27335438 0.74 TRPV1 (0.48) POLQTRPV1HSD11B1HDAC6TSHR
SCHEMBL7968895 0.73 ALDH1A1 (0.43) ALDH1A1MEN1KMT2ANPC1RAB9A
SCHEMBL15206612 0.73 TDP1 (0.51) ALDH1A1TSHRMEN1KMT2AHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6235730-B1 ANTICHOLESTEROL AGENT, ANTILIPEMIC AGENT JAPAN TOBACCO, INC. (JP) 2001-05-22 US disclosed
CN-1252068-A 3-piperidyl-4-oxoquinazoline derivatives and pharmaceutical compositions containing the same JAPAN TOBACCO INC (JP) 2000-05-03 CN disclosed
EP-0970954-A1 3-PIPERIDYL-4-OXOQUINAZOLINE DERIVATIVES AND MEDICINCAL COMPOSITIONS CONTAINING THE SAME JAPAN TOBACCO INC. (JP) 2000-01-12 EP disclosed