SCHEMBL7986402

SCHEMBL7986402

BrCCC(CCBr)c1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 4/20 0.42
HTR2A P28223 5/20 0.40
TDP1 Q9NUW8 1/20 0.40
TAAR1 Q96RJ0 1/20 0.40
GABBR2 O75899 2/20 0.39
GABBR1 Q9UBS5 2/20 0.39
DPP4 P27487 2/20 0.38
TSHR P16473 2/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2D6 P10635 1/20 0.38
PKM P14618 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
TRPA1 O75762 1/20 0.38
ALDH1A1 P00352 1/20 0.38
F2 P00734 1/20 0.38
SIGMAR1 Q99720 1/20 0.38
MTOR P42345 1/20 0.37
RAB9A P51151 1/20 0.37
GRM7 Q14831 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10812162 0.90 HRH1 (0.39) HRH1HTR2ATDP1TAAR1GABBR2
SCHEMBL5478216 0.89 TSHR (0.36) HRH1HTR2ATDP1TAAR1GABBR2
SCHEMBL30312009 0.89 AOC3 (0.42) HRH1HTR2ATAAR1SIGMAR1
SCHEMBL1310414 0.89 TRPA1 (0.44) HRH1HTR2ATDP1TAAR1GABBR2
SCHEMBL6529288 0.86 TRPA1 (0.39) HRH1HTR2ATDP1TAAR1GABBR2
SCHEMBL11566039 0.83 RIPK1 (0.36) HRH1HTR2ATDP1TAAR1GABBR2
SCHEMBL2172475 0.81 HRH1 (0.56) HRH1HTR2ATDP1TAAR1CYP1A2
SCHEMBL30171026 0.79 HRH1 (0.54) HRH1HTR2ATDP1TAAR1CYP1A2
SCHEMBL3683571 0.78 CYP1A2 (0.51) GABBR2GABBR1CYP1A2CYP2D6PKM
SCHEMBL9452584 0.78 HTR2A (0.43) HRH1HTR2ATAAR1GABBR2GABBR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6235731-B1 REDUCING BLOOD LIPIDS, SUGARS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-05-22 US disclosed
EP-0915888-A1 FUSED IMIDAZOPYRIDINE DERIVATIVES AS ANTIHYPERLIPIDEMIC AGENTS Takeda Chemical Industries, Ltd. (JP) 1999-05-19 EP disclosed
WO-1997040051-A1 FUSED IMIDAZOPYRIDINE DERIVATIVES AS ANTIHYPERLIPIDEMIC AGENTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-10-30 WO disclosed