SCHEMBL7986816

SCHEMBL7986816

CC(CN(C)C)Cn1cc(-c2cncc(-c3ccccc3)c2)c2c(Cl)cccc21

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 5/20 0.58
FLT1 P17948 2/20 0.58
FLT4 P35916 2/20 0.58
PRKACA P17612 1/20 0.38
PRKACG P22612 1/20 0.38
PRKACB P22694 1/20 0.38
GRIN2B Q13224 5/20 0.35
SMO Q99835 1/20 0.34
ASH1L Q9NR48 1/20 0.33
KCNH2 Q12809 3/20 0.31
DYRK1A Q13627 1/20 0.31
GRIN1 Q05586 1/20 0.31
PTGDR2 Q9Y5Y4 1/20 0.31
CHRM2 P08172 2/20 0.31
HTR1A P08908 2/20 0.31
ADRA2A P08913 2/20 0.31
CHRM1 P11229 2/20 0.31
DRD1 P21728 2/20 0.31
TBXA2R P21731 2/20 0.31
SLC6A2 P23975 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7554934 0.93 KDR (0.55) KDRFLT1FLT4PRKACAPRKACG
SCHEMBL7504511 0.92 KDR (0.54) KDRFLT1FLT4PRKACAPRKACG
SCHEMBL7551047 0.90 KDR (0.51) KDRFLT1FLT4PRKACAPRKACG
SCHEMBL7552915 0.89 KDR (0.51) KDRFLT1FLT4PRKACAPRKACG
SCHEMBL7987137 0.88 KDR (0.74) KDRFLT1FLT4PRKACAPRKACG
SCHEMBL7550357 0.84 KDR (0.78) KDRFLT1FLT4PRKACAPRKACG
SCHEMBL7548486 0.84 KDR (0.41) KDRFLT1FLT4GRIN2BSMO
SCHEMBL7990966 0.82 KDR (0.63) KDRFLT1FLT4PRKACAPRKACG
SCHEMBL7987886 0.82 KDR (0.63) KDRFLT1FLT4PRKACAPRKACG
SCHEMBL7550081 0.82 KDR (0.56) KDRFLT1FLT4PRKACAPRKACG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6265403-B1 TYROSINE INHIBITORS MERCK & CO., INC. 2001-07-24 US disclosed