SCHEMBL7990966

SCHEMBL7990966

CC(CN(C)C)Cn1cc(-c2cncc(-c3ccccc3)c2)c2ccc(Cl)cc21

nearest known ligand 0.63

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDR P35968 7/20 0.63
FLT1 P17948 4/20 0.63
FLT4 P35916 4/20 0.63
PRKACA P17612 1/20 0.39
PRKACG P22612 1/20 0.39
PRKACB P22694 1/20 0.39
KCNH2 Q12809 2/20 0.38
DYRK1A Q13627 2/20 0.38
HTR6 P50406 1/20 0.37
MDM4 O15151 1/20 0.35
TP53 P04637 1/20 0.35
MDM2 Q00987 1/20 0.35
ASH1L Q9NR48 1/20 0.35
KCNA3 P22001 2/20 0.34
NR1D1 P20393 2/20 0.34
MAT2A P31153 1/20 0.34
IDH1 O75874 1/20 0.34
SCN5A Q14524 1/20 0.33
SCN9A Q15858 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7548685 0.94 KDR (0.60) KDRFLT1FLT4PRKACAPRKACG
SCHEMBL7508525 0.93 KDR (0.59) KDRFLT1FLT4PRKACAPRKACG
SCHEMBL7987886 0.92 KDR (0.63) KDRFLT1FLT4PRKACAPRKACG
SCHEMBL7976518 0.89 KDR (0.72) KDRFLT1FLT4PRKACAPRKACG
SCHEMBL7550357 0.89 KDR (0.78) KDRFLT1FLT4PRKACAPRKACG
SCHEMBL7505482 0.88 KDR (0.54) KDRFLT1FLT4PRKACAPRKACG
SCHEMBL7994231 0.87 KDR (0.70) KDRFLT1FLT4PRKACAPRKACG
SCHEMBL7988018 0.87 KDR (0.78) KDRFLT1FLT4PRKACAPRKACG
SCHEMBL7506521 0.86 KDR (0.60) KDRFLT1FLT4PRKACAPRKACG
SCHEMBL7513664 0.85 KDR (0.59) KDRFLT1FLT4PRKACAPRKACG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6265403-B1 TYROSINE INHIBITORS MERCK & CO., INC. 2001-07-24 US disclosed