SCHEMBL7987209

SCHEMBL7987209

c1ccc(-c2cncc(-c3cn(CCN4CCOCC4)c4cccnc34)c2)cc1

nearest known ligand 0.58

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KDR P35968 4/20 0.58
FLT1 P17948 3/20 0.58
FLT4 P35916 3/20 0.58
GSK3B P49841 3/20 0.50
NFATC1 O95644 1/20 0.45
DYRK1A Q13627 1/20 0.45
CNR1 P21554 1/20 0.42
CNR2 P34972 1/20 0.42
MAPK14 Q16539 1/20 0.41
SLC2A1 P11166 1/20 0.40
TLR9 Q9NR96 1/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7554499 0.91 KDR (0.53) KDRFLT1FLT4GSK3BNFATC1
SCHEMBL7548593 0.91 KDR (0.57) KDRFLT1FLT4GSK3BMAPK14
SCHEMBL7987884 0.89 KDR (0.52) KDRFLT1FLT4GSK3BNFATC1
SCHEMBL7990494 0.88 KDR (0.51) KDRFLT1FLT4GSK3BNFATC1
SCHEMBL7990540 0.87 KDR (0.75) KDRFLT1FLT4GSK3BNFATC1
SCHEMBL7554860 0.87 CYP1A2 (0.49) KDRFLT1FLT4GSK3BNFATC1
SCHEMBL7502516 0.85 KDR (0.77) KDRFLT1FLT4GSK3BNFATC1
SCHEMBL7556924 0.84 KDR (0.59) KDRFLT1FLT4GSK3BNFATC1
SCHEMBL7548014 0.84 KDR (0.43) KDRFLT1FLT4GSK3B
SCHEMBL7547227 0.84 KDR (0.60) KDRFLT1FLT4GSK3BNFATC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6265403-B1 TYROSINE INHIBITORS MERCK & CO., INC. 2001-07-24 US disclosed