SCHEMBL7990540

SCHEMBL7990540

c1cnc2c(-c3cncc(-c4ccsc4)c3)cn(CCN3CCOCC3)c2c1

nearest known ligand 0.75

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KDR P35968 10/20 0.75
FLT1 P17948 5/20 0.75
FLT4 P35916 5/20 0.75
GSK3B P49841 3/20 0.45
NFATC1 O95644 1/20 0.44
DYRK1A Q13627 1/20 0.44
MAPK14 Q16539 1/20 0.40
GAK O14976 1/20 0.40
CYP2A6 P11509 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7993940 0.91 KDR (0.74) KDRFLT1FLT4GSK3BMAPK14
SCHEMBL7987209 0.87 KDR (0.58) KDRFLT1FLT4GSK3BNFATC1
SCHEMBL7990489 0.86 KDR (0.75) KDRFLT1FLT4GSK3BNFATC1
SCHEMBL7549006 0.86 KDR (0.75) KDRFLT1FLT4GSK3BNFATC1
SCHEMBL7557708 0.86 KDR (0.56) KDRFLT1FLT4GSK3BNFATC1
SCHEMBL7506453 0.85 KDR (1.00) KDRFLT1FLT4GSK3BNFATC1
SCHEMBL7554499 0.85 KDR (0.53) KDRFLT1FLT4GSK3BNFATC1
SCHEMBL7987884 0.83 KDR (0.52) KDRFLT1FLT4GSK3BNFATC1
SCHEMBL7990494 0.82 KDR (0.51) KDRFLT1FLT4GSK3BNFATC1
SCHEMBL7990322 0.82 KDR (0.73) KDRFLT1FLT4GSK3BNFATC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6265403-B1 TYROSINE INHIBITORS MERCK & CO., INC. 2001-07-24 US disclosed