SCHEMBL7987814

SCHEMBL7987814

O=c1[nH]c2ccc3c(c2[nH]c1=O)CNCC3

nearest known ligand 0.77

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
GRIA1 P42261 1/20 0.50
GRIA2 P42262 1/20 0.50
GRIA3 P42263 1/20 0.50
GRIA4 P48058 1/20 0.50
PNMT P11086 4/20 0.45
ADRA2A P08913 1/20 0.45
ADRA2B P18089 1/20 0.45
ADRA2C P18825 1/20 0.45
PARP1 P09874 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6780495 0.87 GRIA1 (0.50) GRIA1GRIA2GRIA3GRIA4PNMT
SCHEMBL9091481 0.77 GRIA1 (0.58) GRIA1GRIA2GRIA3GRIA4
SCHEMBL29850336 0.72 PNMT (0.46) PNMTADRA2AADRA2BADRA2CPARP1
SCHEMBL6780272 0.71 GRIA1 (0.45) GRIA1GRIA2GRIA3GRIA4
SCHEMBL6786694 0.70 GRIA1 (0.53) GRIA1GRIA2GRIA3GRIA4
SCHEMBL8670950 0.70 GRIA1 (0.43) GRIA1GRIA2GRIA3GRIA4
SCHEMBL7617146 0.69 PNMT (0.49) PNMTADRA2AADRA2BADRA2C
Hydrochloric Acid SCHEMBL6785550 0.69 GRIA1 (0.52) GRIA1GRIA2GRIA3GRIA4
SCHEMBL6780845 0.67 GRIA1 (0.56) GRIA1GRIA2GRIA3GRIA4PNMT
SCHEMBL7983799 0.67 GRIA1 (0.60) GRIA1GRIA2GRIA3GRIA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6197771-B1 NERVOUS SYSTEM DISORDERS; ANTIISCHEMIC AGENTS; ALZHEIMER'SDISEASE; PARKINSON'S DISEASE; HUNTINGTON'S DISEASE WARNER-LAMBERT COMPANY 2001-03-06 US disclosed
US-6057313-A TREATING CENTRAL NERVOUS SYSTEM DISORDERS WARNER-LAMBERT COMPANY (US) 2000-05-02 US disclosed
WO-1996028445-A1 NOVEL GLUTAMATE (AMPA/KAINATE) RECEPTOR ANTAGONISTS: N-SUBSTITUTED FUSED AZACYCLOALKYLQUINOXALINEDIONES WARNER-LAMBERT COMPANY (US) 1996-09-19 WO disclosed