SCHEMBL7987876

SCHEMBL7987876

COc1ccc2c(c1)c(-c1cncc(-c3ccc(Cl)cc3)c1)cn2C(C)CN(C)C

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 2/20 0.45
PDE4D Q08499 2/20 0.45
HTR6 P50406 3/20 0.41
CYP11B1 P15538 5/20 0.38
CYP11B2 P19099 5/20 0.38
CYP17A1 P05093 4/20 0.38
FLT1 P17948 1/20 0.37
FLT4 P35916 1/20 0.37
KDR P35968 1/20 0.37
ALPL P05186 2/20 0.37
CYP3A4 P08684 1/20 0.36
AKR1C3 P42330 2/20 0.35
AKR1C4 P17516 1/20 0.35
PTGS1 P23219 1/20 0.35
AKR1C2 P52895 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7549809 0.94 HTR6 (0.43) PDE4BPDE4DHTR6CYP11B1CYP11B2
SCHEMBL7555466 0.90 PDE4B (0.46) PDE4BPDE4DHTR6CYP11B1CYP11B2
SCHEMBL7990227 0.90 PDE4B (0.45) PDE4BPDE4DHTR6CYP11B1CYP11B2
SCHEMBL7990418 0.89 KDR (0.39) PDE4BPDE4DCYP11B1CYP11B2CYP17A1
SCHEMBL7976435 0.88 PRKCA (0.42) PDE4BPDE4DHTR6CYP11B1CYP11B2
SCHEMBL7550632 0.87 PDE4B (0.43) PDE4BPDE4DHTR6CYP11B1CYP11B2
SCHEMBL7550587 0.85 KDR (0.49) PDE4BPDE4DHTR6CYP11B1CYP11B2
SCHEMBL7552885 0.85 KDR (0.51) PDE4BPDE4DHTR6FLT1FLT4
SCHEMBL7516192 0.85 KDR (0.54) PDE4BPDE4DHTR6CYP11B1CYP11B2
SCHEMBL7991178 0.85 KDR (0.54) PDE4BPDE4DHTR6FLT1FLT4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6265403-B1 TYROSINE INHIBITORS MERCK & CO., INC. 2001-07-24 US disclosed