Nimetazepam

Nimetazepam

SCHEMBL79886

CN1C(=O)CN=C(c2ccccc2)c2cc([N+](=O)[O-])ccc21

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 1.00
GABRA1 P14867 8/20 0.76
GABRG2 P18507 8/20 0.76
GABRB3 P28472 8/20 0.76
GABRA5 P31644 8/20 0.76
GABRA3 P34903 8/20 0.76
GABRA2 P47869 7/20 0.74
GABRB2 P47870 5/20 0.74
OPRK1 P41145 2/20 0.74
CCKBR P32239 2/20 0.74
MC3R P41968 1/20 0.74
GHSR Q92847 1/20 0.74
GABRP O00591 1/20 0.67
GABRD O14764 1/20 0.67
CACNA1F O60840 1/20 0.67
ALB P02768 1/20 0.67
GABRB1 P18505 1/20 0.67
AKR1C3 P42330 1/20 0.67
GABRA4 P48169 1/20 0.67
AKR1C2 P52895 1/20 0.67

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Nimetazepam SCHEMBL29374297 1.00 LMNA (1.00) LMNAGABRA1GABRG2GABRB3GABRA5
Nimetazepam SCHEMBL10689471 0.98 LMNA (0.95) LMNAGABRA1GABRG2GABRB3GABRA5
Nimetazepam SCHEMBL9542099 0.98 LMNA (0.95) LMNAGABRA1GABRG2GABRB3GABRA5
Nimetazepam SCHEMBL1003526 0.90 LMNA (0.81) LMNAGABRA1GABRG2GABRB3GABRA5
SCHEMBL18319288 0.88 LMNA (0.79) LMNAGABRA1GABRG2GABRB3GABRA5
SCHEMBL5044330 0.88 LMNA (0.78) LMNAGABRA1GABRG2GABRB3GABRA5
Flunitrazepam SCHEMBL1900353 0.87 GABRA1 (0.80) LMNAGABRA1GABRG2GABRB3GABRA5
Flunitrazepam SCHEMBL8812488 0.85 GABRA1 (1.00) LMNAGABRA1GABRG2GABRB3GABRA5
SCHEMBL9473650 0.85 GABRA1 (0.78) LMNAGABRA1GABRG2GABRB3GABRA5
Flunitrazepam SCHEMBL44169 0.85 GABRA1 (1.00) LMNAGABRA1GABRG2GABRB3GABRA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 3953 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260076953-A1 METHODS OF DIAGNOSING AND TREATING ADHD IN BIOMARKER POSITIVE SUBJECTS THE CHILDREN'S HOSPITAL OF PHILADELPHIA (US) 2026-03-19 US claimed
EP-3507371-B1 COMPOSITIONS FOR TREATING DISEASES AND DISORDERS OF THE NERVOUS SYSTEM UNIV RUTGERS (US) 2026-01-28 EP claimed
US-20250375421-A1 METHODS OF USING DMT SHULMAN WILLIAM (US) 2025-12-11 US claimed
US-12396981-B2 Methods of using DMT SHULMAN WILLIAM (US) 2025-08-26 US claimed
US-12350379-B2 Extended release pharmaceutical formulation and methods of treatment DOUGLAS PHARMACETICALS LTD (NZ) 2025-07-08 US claimed
US-20250120962-A1 NONSELECTIVE METABOTROPIC GLUTAMATE RECEPTOR ACTIVATORS FOR TREATMENT OF ATTENTION DEFICIT DISORDER AND 22Q SYNDROME THE CHILDREN'S HOSPITAL OF PHILADELPHIA (US) 2025-04-17 US claimed
EP-3518975-B1 FORMULATION COMPRISING FENFLURAMINE AND CANNABIDIOL AND ITS USE IN THE TREATMENT OF SEIZURES ZOGENIX INTERNATIONAL LTD (GB) 2025-04-09 EP claimed
EP-4023222-B1 NONSELECTIVE METABOTROPIC GLUTAMATE RECEPTOR ACTIVATOR FOR TREATMENT OF 22Q SYNDROME CHILDRENS HOSPITAL PHILADELPHIA (US) 2024-12-18 EP claimed
US-12133922-B2 Abuse resistant capsule R.P. SCHERER TECHNOLOGIES, LLC (US) 2024-11-05 US claimed
US-20240307386-A1 NOVEL METHODS INTRA-CELLULAR THERAPIES, INC. 2024-09-19 US claimed
EP-0233276-A4 WRAPPING. CROWELL CORP (US) 1988-12-15 EP claimed
EP-0281324-A2 Improved passivation for integrated circuit structures ADVANCED MICRO DEVICES, INC. (US) 1988-09-07 EP claimed
US-4721709-A Novel pharmaceutical compositions containing hydrophobic practically water-insoluble drugs adsorbed on pharmaceutical excipients as carrier; process for their preparation and the use of said compositions PYARE SETH (CH) 1988-01-26 US claimed
EP-0233276-A1 WRAPPING. CROWELL CORP (US) 1987-08-26 EP claimed
WO-1987001092-A1 WRAPPING THE CROWELL CORPORATION (US) 1987-02-26 WO claimed
US-4557934-A ALONG WITH A DIOL PYRROLIDONE OR AN AZACYCLOPENTAN-2-ONE THE PROCTER & GAMBLE COMPANY (US) 1985-12-10 US claimed
EP-0153939-A1 VACCINE AND ANTIGEN AGAINST PALUDISM AND PREPARATION PROCESS THEREOF INSTITUT MERIEUX (FR) 1985-09-11 EP claimed
WO-1985000977-A1 VACCINE AND ANTIGEN AGAINST PALUDISM AND PREPARATION PROCESS THEREOF INSTITUT MERIEUX S.A. (FR) 1985-03-14 WO claimed
EP-0010899-B1 PROCESS FOR CONCENTRATING DILUTE SULPHURIC ACID IN AN EVAPORATOR AIR PRODUCTS AND CHEMICALS, INC. (US) 1983-02-02 EP claimed
US-4044003-A Process for preparing 1,4-benzodiazepines SUMITOMO CHEMICAL COMPANY, LIMITED (JA) 1977-08-23 US claimed