Nimetazepam

Nimetazepam

SCHEMBL1003526

CN1C(=O)CN=C(c2ccccc2)c2cc([N+](=O)[O-])ccc21.O=C1CN=C(c2ccccc2)c2cc([N+](=O)[O-])ccc2N1

nearest known ligand 0.81

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.81
PDE4D Q08499 2/20 0.77
HPGD P15428 1/20 0.77
GABRA1 P14867 10/20 0.63
GABRG2 P18507 10/20 0.63
GABRB3 P28472 10/20 0.63
GABRA5 P31644 10/20 0.63
GABRA3 P34903 10/20 0.63
GABRA2 P47869 9/20 0.62
GABRB2 P47870 7/20 0.62
OPRK1 P41145 3/20 0.62
CCKBR P32239 2/20 0.62
MC3R P41968 1/20 0.62
GHSR Q92847 1/20 0.62
CHRM1 P11229 1/20 0.60
GABRP O00591 2/20 0.58
GABRD O14764 2/20 0.58
GABRB1 P18505 2/20 0.58
GABRA4 P48169 2/20 0.58
GABRE P78334 2/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Flunitrazepam SCHEMBL28086646 0.93 GABRA1 (0.75) LMNAPDE4DHPGDGABRA1GABRG2
Clonazepam SCHEMBL17728660 0.90 GABRA1 (0.67) LMNAPDE4DHPGDGABRA1GABRG2
Nimetazepam SCHEMBL29374297 0.90 LMNA (1.00) LMNAPDE4DHPGDGABRA1GABRG2
Nimetazepam SCHEMBL79886 0.90 LMNA (1.00) LMNAPDE4DHPGDGABRA1GABRG2
Nimetazepam SCHEMBL10689471 0.88 LMNA (0.95) LMNAPDE4DHPGDGABRA1GABRG2
Nimetazepam SCHEMBL9542099 0.88 LMNA (0.95) LMNAPDE4DHPGDGABRA1GABRG2
Nitrazepam SCHEMBL35202 0.88 PDE4D (1.00) LMNAPDE4DHPGDGABRA1GABRG2
Nitrazepam SCHEMBL9747297 0.88 PDE4D (1.00) LMNAPDE4DHPGDGABRA1GABRG2
Nitrazepam SCHEMBL29408437 0.88 PDE4D (1.00) LMNAPDE4DHPGDGABRA1GABRG2
Flunitrazepam SCHEMBL8364961 0.86 GABRA1 (0.64) LMNAPDE4DHPGDGABRA1GABRG2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593104-A2 METHODS OF TREATING AND PREVENTING/REDUCING THE LIKELIHOOD OF MESIAL TEMPORAL LOBE EPILEPSY (TLE) Müller, Prof. Dr., Wolfgang (DE) 2013-05-22 EP disclosed
WO-2011011692-A2 METHODS OF TREATING AND PREVENTING/REDUCING THE LIKELIHOOD OF MESIAL TEMPORAL LOBE EPILEPSY (TLE) STC.UNM (US) 2011-01-27 WO disclosed