SCHEMBL7989587

SCHEMBL7989587

CCOC(=O)Cn1nc2c(c1OC)CN(C(=O)OC(C)(C)C)CC2

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 2/20 0.46
C5AR1 P21730 6/20 0.41
F12 P00748 1/20 0.40
MAPT P10636 3/20 0.39
MTOR P42345 2/20 0.38
ESR2 Q92731 1/20 0.36
KDM4E B2RXH2 1/20 0.36
NR1H2 P55055 1/20 0.35
AKR1B10 O60218 1/20 0.35
AKR1B1 P15121 1/20 0.35
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7992630 0.88 ADORA1 (0.46) ADORA1C5AR1F12MAPTMTOR
SCHEMBL1007338 0.77 TRPM2 (0.45) ADORA1MAPTCYP2C19
SCHEMBL31700101 0.77 ADORA1 (0.51) ADORA1C5AR1F12MAPTMTOR
SCHEMBL22716373 0.76 ADORA1 (0.43) ADORA1C5AR1F12MAPTMTOR
SCHEMBL1885657 0.76 F12 (0.57) ADORA1C5AR1F12MAPTESR2
SCHEMBL22718671 0.76 ADORA1 (0.46) ADORA1C5AR1F12MAPTMTOR
SCHEMBL7988759 0.75 KMT2A (0.50) ADORA1C5AR1MAPTESR2NR1H2
SCHEMBL31700014 0.75 ADORA1 (0.49) ADORA1C5AR1F12MAPTMTOR
SCHEMBL7975140 0.75 ESR2 (0.44) ADORA1MAPTESR2NR1H2
SCHEMBL1007022 0.75 ADORA1 (0.45) ADORA1MAPTCYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6265418-B1 ANTICOAGULANTS UBE INDUSTRIES, LTD. (JP) 2001-07-24 US disclosed
EP-1020467-A1 N-ACYLAMINO ACID AMIDE COMPOUNDS AND INTERMEDIATES FOR PREPARATION THEREOF UBE INDUSTRIES LIMITED (JP) 2000-07-19 EP disclosed