SCHEMBL7989806

SCHEMBL7989806

CCCCc1nc(C[C@H](C(=O)N[C@@H](Cc2cccc3ccccc23)C(=O)O)c2ccc3c(c2)OCO3)cn1C(=O)OC(C)(C)C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EDNRA P25101 4/20 0.40
CTSS P25774 1/20 0.38
CTSK P43235 1/20 0.38
MME P08473 1/20 0.37
ACE P12821 1/20 0.37
CPA1 P15085 1/20 0.37
ACE2 Q9BYF1 1/20 0.37
ITGB3 P05106 2/20 0.37
ITGAV P06756 2/20 0.37
ITGA2B P08514 2/20 0.37
ITGB5 P18084 1/20 0.37
CCKAR P32238 2/20 0.35
CCKBR P32239 2/20 0.35
OPRD1 P41143 2/20 0.35
HRH4 Q9H3N8 1/20 0.34
MAPT P10636 2/20 0.34
CYP3A4 P08684 2/20 0.34
ALDH1A1 P00352 2/20 0.34
LMNA P02545 1/20 0.34
PTGFR P43088 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7989999 0.93 EDNRA (0.40) EDNRACTSSCTSKACEITGB3
SCHEMBL7976826 0.91 MAPK1 (0.45) CTSSCTSKACE
SCHEMBL7986462 0.89 MAPK1 (0.44) CTSSCTSKACE
SCHEMBL8807798 0.86 MAPK1 (0.46) CTSSCTSKACE
SCHEMBL7986434 0.85 EDNRA (0.41) EDNRAITGB3ITGAVITGA2BITGB5
SCHEMBL7988163 0.84 SMN1; SMN2 (0.44) MAPTLMNA
SCHEMBL7990508 0.84 SMN1; SMN2 (0.44) MAPTLMNA
SCHEMBL7990070 0.84 MAPK1 (0.47) CTSSCTSKACE
SCHEMBL7994280 0.84 TACR1 (0.46)
SCHEMBL7994192 0.83 EDNRA (0.41) EDNRAITGB3ITGAVITGA2BITGB5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6207686-B1 FOR THERAPY OF HYPERTENSION FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-03-27 US disclosed
WO-1996015109-A1 ENDOTHELIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1996-05-23 WO disclosed