SCHEMBL7990044

SCHEMBL7990044

Cc1cccc(N2CCN(CCc3ccccc3)CC2)c1

nearest known ligand 0.72

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.72
HTR1A P08908 1/20 0.71
DRD2 P14416 1/20 0.71
MAPT P10636 1/20 0.71
NPSR1 Q6W5P4 1/20 0.71
SIGMAR1 Q99720 5/20 0.70
OPRM1 P35372 1/20 0.59
HRH3 Q9Y5N1 1/20 0.59
ADRA1D P25100 1/20 0.58
ADRA1A P35348 1/20 0.58
ADRA1B P35368 1/20 0.58
MEN1 O00255 1/20 0.58
ALDH1A1 P00352 1/20 0.58
KMT2A Q03164 1/20 0.58
HTR7 P34969 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15961301 0.92 KCNH2 (0.77) KCNH2HTR1ADRD2MAPTNPSR1
SCHEMBL7995650 0.91 HTR1A (0.71) KCNH2HTR1ADRD2MAPTNPSR1
SCHEMBL11560357 0.87 MAPT (0.67) KCNH2HTR1ADRD2MAPTNPSR1
Hydrochloric Acid SCHEMBL3712573 0.86 MAPT (0.75) KCNH2HTR1ADRD2MAPTNPSR1
SCHEMBL13711972 0.86 KCNH2 (0.84) KCNH2DRD2HTR7
SCHEMBL6509439 0.84 DRD2 (1.00) KCNH2HTR1ADRD2MAPTNPSR1
SCHEMBL4523970 0.84 KCNH2 (1.00) KCNH2SIGMAR1HTR7
SCHEMBL13501370 0.84 HTR1A (0.73) HTR1ADRD2MAPTNPSR1SIGMAR1
SCHEMBL9373313 0.82 SIGMAR1 (1.00) KCNH2HTR1ADRD2SIGMAR1HTR7
SCHEMBL4519876 0.81 KCNH2 (1.00) KCNH2HTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6313297-B1 CATALYTIC ALKYLATION; BY-PRODUCT INHIBITION AVENTIS RESEARCH & TECHNOLOGIES (DE) 2001-11-06 US disclosed
EP-1047680-A2 BASE-CATALYZED SYNTHESIS OF 1-ARYL-4-(ARYL ETHYL)PIPERAZINES FROM AROMATIC OLEFINS AND 1-ARYL PIPERAZINES Aventis Research & Technologies GmbH & Co KG (DE) 2000-11-02 EP disclosed
WO-1999036412-A2 BASE-CATALYZED SYNTHESIS OF 1-ARYL-4-(ARYL ETHYL)PIPERAZINES FROM AROMATIC OLEFINS AND 1-ARYL PIPERAZINES AVENTIS RESEARCH & TECHNOLOGIES GMBH & CO. KG (DE) 1999-07-22 WO disclosed