SCHEMBL7990490

SCHEMBL7990490

COc1cccc2c(-c3cncc(-c4cccc(Cl)c4)c3)cn(CCN3CCOCC3)c12

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 3/20 0.49
FLT1 P17948 1/20 0.49
FLT4 P35916 1/20 0.49
PDE4B Q07343 1/20 0.48
CNR2 P34972 9/20 0.44
MAPK13 O15264 1/20 0.42
MAPK12 P53778 1/20 0.42
MAPK11 Q15759 1/20 0.42
MAPK14 Q16539 1/20 0.42
GSK3B P49841 2/20 0.41
CNR1 P21554 2/20 0.40
PTGER2 P43116 1/20 0.40
MEN1 O00255 1/20 0.40
LMNA P02545 1/20 0.40
MAPT P10636 1/20 0.40
KMT2A Q03164 1/20 0.40
NFATC1 O95644 1/20 0.40
DYRK1A Q13627 1/20 0.40
TNIK Q9UKE5 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7550092 0.92 KDR (0.49) KDRFLT1FLT4PDE4BCNR2
SCHEMBL7990572 0.92 KDR (0.50) KDRFLT1FLT4PDE4BCNR2
SCHEMBL7990350 0.91 KDR (0.55) KDRFLT1FLT4CNR2GSK3B
SCHEMBL7976879 0.90 KDR (0.50) KDRFLT1FLT4CNR2GSK3B
SCHEMBL7987655 0.87 KDR (0.51) KDRFLT1FLT4CNR2GSK3B
SCHEMBL7553648 0.87 KDR (0.50) KDRFLT1FLT4CNR2MAPK13
SCHEMBL7549301 0.87 KDR (0.52) KDRFLT1FLT4CNR2MAPK13
SCHEMBL7550496 0.87 CNR2 (0.38) KDRFLT1FLT4PDE4BCNR2
SCHEMBL7987725 0.85 KDR (0.70) KDRFLT1FLT4CNR2GSK3B
SCHEMBL7554271 0.84 KDR (0.49) KDRFLT1FLT4CNR2GSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6265403-B1 TYROSINE INHIBITORS MERCK & CO., INC. 2001-07-24 US disclosed