SCHEMBL7987725

SCHEMBL7987725

COc1cccc2c(-c3cncc(-c4ccsc4)c3)cn(CCN3CCOCC3)c12

nearest known ligand 0.70

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KDR P35968 10/20 0.70
FLT1 P17948 4/20 0.70
FLT4 P35916 4/20 0.70
CNR2 P34972 8/20 0.43
GSK3B P49841 2/20 0.42
NFATC1 O95644 1/20 0.41
DYRK1A Q13627 1/20 0.41
CNR1 P21554 2/20 0.40
CYP2D6 P10635 1/20 0.38
TSHR P16473 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7990673 0.92 KDR (0.69) KDRFLT1FLT4CNR2
SCHEMBL7990350 0.88 KDR (0.55) KDRFLT1FLT4CNR2GSK3B
SCHEMBL7554218 0.88 KDR (0.71) KDRFLT1FLT4CNR2GSK3B
SCHEMBL7993934 0.87 KDR (0.70) KDRFLT1FLT4CNR2GSK3B
SCHEMBL7547303 0.87 KDR (0.53) KDRFLT1FLT4CNR2CNR1
SCHEMBL7987655 0.86 KDR (0.51) KDRFLT1FLT4CNR2GSK3B
SCHEMBL7990572 0.86 KDR (0.50) KDRFLT1FLT4CNR2GSK3B
SCHEMBL7976879 0.86 KDR (0.50) KDRFLT1FLT4CNR2GSK3B
SCHEMBL7990490 0.85 KDR (0.49) KDRFLT1FLT4CNR2GSK3B
SCHEMBL7506453 0.82 KDR (1.00) KDRFLT1FLT4CNR2GSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6265403-B1 TYROSINE INHIBITORS MERCK & CO., INC. 2001-07-24 US disclosed