SCHEMBL7990512

SCHEMBL7990512

O=C(O)Cc1ccc2c(c1)OCC(Cc1ccccc1)O2

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LTB4R Q15722 2/20 0.59
LTB4R2 Q9NPC1 2/20 0.59
HTT P42858 1/20 0.50
AIMP2 Q13155 4/20 0.47
POLB P06746 2/20 0.47
AKR1B1 P15121 1/20 0.47
HPGD P15428 3/20 0.46
CYP1A2 P05177 2/20 0.46
CYP2D6 P10635 2/20 0.46
CYP2C9 P11712 2/20 0.46
CYP2C19 P33261 2/20 0.46
ALDH1A1 P00352 3/20 0.46
MEN1 O00255 1/20 0.46
LMNA P02545 1/20 0.46
KMT2A Q03164 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.45
DRD2 P14416 1/20 0.45
DRD4 P21917 1/20 0.45
DRD3 P35462 1/20 0.45
ALOX5 P09917 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10389548 0.85 LTB4R (0.47) LTB4RLTB4R2HTTAIMP2POLB
SCHEMBL14053644 0.78 LTB4R (0.48) LTB4RLTB4R2HTTAIMP2POLB
SCHEMBL8785209 0.74 LTB4R (1.00) LTB4RLTB4R2
SCHEMBL8785623 0.74 LTB4R (1.00) LTB4RLTB4R2
SCHEMBL8785049 0.74 LTB4R (1.00) LTB4RLTB4R2
SCHEMBL8785213 0.74 LTB4R (1.00) LTB4RLTB4R2
SCHEMBL10387689 0.73 CYP3A4 (0.51) LTB4RLTB4R2HTTPOLBAKR1B1
SCHEMBL22068562 0.72 CA2 (0.53) LMNASMN1; SMN2DRD2DRD4DRD3
SCHEMBL29642680 0.72 CYP3A4 (0.75) HPGDCYP1A2CYP2D6CYP2C19ALDH1A1
SCHEMBL286952 0.72 ALDH1A1 (0.60) HTTAKR1B1HPGDCYP1A2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6207686-B1 FOR THERAPY OF HYPERTENSION FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-03-27 US disclosed
EP-0792265-A1 ENDOTHELIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-09-03 EP disclosed
WO-1996015109-A1 ENDOTHELIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1996-05-23 WO disclosed