Morpholine

Morpholine

SCHEMBL7990935

C1COCCN1.CCC(SC)n1c(-c2ccccc2CN2CCOCC2)nc(-c2ccc(F)cc2)c1-c1ccncc1.CCCn1c(-c2ccc(S(C)(=O)=O)cc2)nc(-c2ccc(F)cc2)c1-c1ccncc1

nearest known ligand 0.37

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 11/20 0.37
MAPK11 Q15759 8/20 0.37
MAPK13 O15264 7/20 0.37
MAPK12 P53778 7/20 0.37
ADORA2A P29274 1/20 0.35
ADORA1 P30542 1/20 0.35
RIPK3 Q9Y572 1/20 0.34
ALOX5 P09917 3/20 0.33
IDO1 P14902 1/20 0.32
GCGR P47871 2/20 0.32
CYP3A4 P08684 2/20 0.32
HSD17B10 Q99714 2/20 0.32
ALDH1A1 P00352 2/20 0.32
CSNK1A1 P48729 1/20 0.32
CSNK1D P48730 1/20 0.32
CSNK1E P49674 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
CSNK1A1L Q8N752 1/20 0.32
CTDSP1 Q9GZU7 1/20 0.31
KDM4E B2RXH2 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5082085 0.85 MAPK14 (0.45) MAPK14MAPK11MAPK13MAPK12ADORA2A
Morpholine SCHEMBL4553714 0.82 MAPK14 (0.49) MAPK14MAPK11MAPK13MAPK12RIPK3
Morpholine SCHEMBL7387653 0.78 MAPK14 (0.39) MAPK14MAPK11MAPK13MAPK12RIPK3
SCHEMBL4566366 0.78 ADORA2A (0.46) MAPK14MAPK11MAPK13MAPK12ADORA2A
Morpholine SCHEMBL7419803 0.74 MAPK14 (0.47) MAPK14MAPK11MAPK13MAPK12RIPK3
SCHEMBL4553711 0.74 MAPK14 (0.55) MAPK14MAPK11MAPK13MAPK12
SCHEMBL7360193 0.74 MAPK14 (0.55) MAPK14MAPK11MAPK13MAPK12
SCHEMBL7232352 0.74 MAPK14 (0.44) MAPK14MAPK11MAPK13MAPK12ADORA2A
SCHEMBL8524296 0.73 MAPK14 (0.46) MAPK14MAPK11MAPK13MAPK12ALOX5
Morpholine SCHEMBL7382870 0.72 ALOX5 (0.40) MAPK14MAPK11MAPK13MAPK12RIPK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6288089-B1 ADMINISTERING A COMPOSITION OF PYRIDYL IMIDAZOLE COMPOUNDS TO TREAT PARKINSON'S DISEASE, HUNTINGTON'S DISEASE, ALZHEIMER'S DISEASE, AND AMYOTOPHIC LATERAL SCLEROSIS NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2001-09-11 US claimed