SCHEMBL7548685

SCHEMBL7548685

CC(CN(C)C)Cn1cc(-c2cncc(-c3ccc(Cl)cc3)c2)c2ccc(Cl)cc21

nearest known ligand 0.60

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KDR P35968 6/20 0.60
FLT1 P17948 3/20 0.60
FLT4 P35916 3/20 0.60
KCNH2 Q12809 1/20 0.39
DYRK1A Q13627 1/20 0.39
PRKACA P17612 1/20 0.37
PRKACG P22612 1/20 0.37
PRKACB P22694 1/20 0.37
SCN5A Q14524 2/20 0.34
SCN9A Q15858 2/20 0.34
NR1D1 P20393 4/20 0.33
MAP4K4 O95819 1/20 0.33
HTR6 P50406 1/20 0.32
IDH1 O75874 1/20 0.31
RAB9A P51151 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7990966 0.94 KDR (0.63) KDRFLT1FLT4KCNH2DYRK1A
SCHEMBL7506521 0.92 KDR (0.60) KDRFLT1FLT4KCNH2DYRK1A
SCHEMBL7508525 0.91 KDR (0.59) KDRFLT1FLT4KCNH2DYRK1A
SCHEMBL7976518 0.91 KDR (0.72) KDRFLT1FLT4KCNH2DYRK1A
SCHEMBL7988018 0.88 KDR (0.78) KDRFLT1FLT4KCNH2DYRK1A
SCHEMBL7505482 0.86 KDR (0.54) KDRFLT1FLT4KCNH2DYRK1A
SCHEMBL7987886 0.86 KDR (0.63) KDRFLT1FLT4KCNH2DYRK1A
SCHEMBL7516192 0.84 KDR (0.54) KDRFLT1FLT4KCNH2HTR6
SCHEMBL7553739 0.84 KDR (0.54) KDRFLT1FLT4KCNH2DYRK1A
SCHEMBL7976277 0.83 KDR (0.43) KDRFLT1FLT4KCNH2DYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1147107-A4 NOVEL ANGIOGENESIS INHIBITORS MERCK & CO INC (US) 2002-05-22 EP claimed
EP-1147107-A1 NOVEL ANGIOGENESIS INHIBITORS Merck & Co., Inc. (US) 2001-10-24 EP claimed
WO-2000043393-A1 NOVEL ANGIOGENESIS INHIBITORS MERCK & CO., INC. (US) 2000-07-27 WO claimed
EP-1147107-A4 NOVEL ANGIOGENESIS INHIBITORS MERCK & CO INC (US) 2002-05-22 EP disclosed
EP-1147107-A1 NOVEL ANGIOGENESIS INHIBITORS Merck & Co., Inc. (US) 2001-10-24 EP disclosed
US-6265403-B1 TYROSINE INHIBITORS MERCK & CO., INC. 2001-07-24 US disclosed
WO-2000043393-A1 NOVEL ANGIOGENESIS INHIBITORS MERCK & CO., INC. (US) 2000-07-27 WO disclosed