SCHEMBL7990969

SCHEMBL7990969

COc1cccc2c(-c3cncc(-c4ccc(Cl)cc4)c3)cn(C(C)C3CCCNC3)c12

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 1/20 0.38
LCK P06239 1/20 0.38
LYN P07948 1/20 0.38
BLK P51451 1/20 0.38
CDK7 P50613 3/20 0.38
CCNH P51946 3/20 0.38
MNAT1 P51948 3/20 0.38
CCNT1 O60563 2/20 0.38
CDK9 P50750 2/20 0.38
CCNE1 P24864 1/20 0.38
CDK2 P24941 1/20 0.38
KCNH2 Q12809 3/20 0.35
SLC6A2 P23975 4/20 0.35
SLC6A4 P31645 4/20 0.35
SLC6A3 Q01959 4/20 0.35
CYP2D6 P10635 2/20 0.35
TLR9 Q9NR96 1/20 0.35
TLR8 Q9NR97 1/20 0.35
TLR7 Q9NYK1 1/20 0.35
ACP1 P24666 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7976911 0.93 TNF (0.36) EGFRLCKLYNBLKCDK7
SCHEMBL7990894 0.92 EGFR (0.42) EGFRLCKLYNBLKCDK7
SCHEMBL7977291 0.92 EGFR (0.38) EGFRLCKLYNBLKCDK7
SCHEMBL7987981 0.88 EGFR (0.38) EGFRLCKLYNBLKKCNH2
SCHEMBL7994041 0.87 KDR (0.41) EGFRLCKLYNBLKCDK7
SCHEMBL7990169 0.84 PDE4B (0.37) CDK7CCNHMNAT1CCNT1CDK9
SCHEMBL7987644 0.83 CCNT1 (0.40) CDK7CCNHMNAT1CCNT1CDK9
SCHEMBL7986838 0.83 CCNT1 (0.40) CDK7CCNHMNAT1CCNT1CDK9
SCHEMBL7976151 0.82 CCNT1 (0.37) CDK7CCNHMNAT1CCNT1CDK9
SCHEMBL7991016 0.82 CCNT1 (0.37) EGFRLCKLYNBLKCDK7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6265403-B1 TYROSINE INHIBITORS MERCK & CO., INC. 2001-07-24 US disclosed