SCHEMBL7987981

SCHEMBL7987981

COc1cccc(-c2cncc(-c3cn(C(C)C4CCCNC4)c4c(OC)cccc34)c2)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 2/20 0.38
LCK P06239 1/20 0.38
LYN P07948 1/20 0.38
BLK P51451 1/20 0.38
CHEK1 O14757 3/20 0.38
CYP2C19 P33261 1/20 0.36
ACP1 P24666 1/20 0.36
KCNH2 Q12809 1/20 0.35
CHRNB4 P30926 1/20 0.35
CHRNA3 P32297 1/20 0.35
EED O75530 1/20 0.35
ABL1 P00519 1/20 0.35
SRC P12931 1/20 0.35
ABL2 P42684 1/20 0.35
CYP11B1 P15538 1/20 0.35
CYP11B2 P19099 1/20 0.35
AXL P30530 1/20 0.34
FLT3 P36888 1/20 0.34
TYRO3 Q06418 1/20 0.34
MERTK Q12866 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7990894 0.92 EGFR (0.42) EGFRLCKLYNBLKCHEK1
SCHEMBL7977291 0.92 EGFR (0.38) EGFRLCKLYNBLKKCNH2
SCHEMBL7976911 0.91 TNF (0.36) EGFRLCKLYNBLKACP1
SCHEMBL7976272 0.90 CCNT1 (0.41) EGFRCHEK1CYP2C19ACP1EED
SCHEMBL7990969 0.88 EGFR (0.38) EGFRLCKLYNBLKACP1
SCHEMBL7975970 0.88 HTR6 (0.39) EGFRLCKLYNBLKCHEK1
SCHEMBL7994041 0.87 KDR (0.41) EGFRLCKLYNBLKCHEK1
SCHEMBL7994923 0.85 PRKCA (0.40) EGFRCHEK1CYP2C19ACP1CHRNB4
SCHEMBL7990984 0.85 CCNT1 (0.36) EGFRLCKLYNBLKCHEK1
SCHEMBL7990463 0.84 CHEK1 (0.39) CHEK1CYP2C19ACP1EED

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6265403-B1 TYROSINE INHIBITORS MERCK & CO., INC. 2001-07-24 US disclosed