SCHEMBL7991453

SCHEMBL7991453

CCCCCOc1cc2c(cc1OC)C(C(=O)c1ccccc1)=NCC2

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.51
HPGD P15428 1/20 0.51
KMT2A Q03164 2/20 0.46
HSD17B10 Q99714 1/20 0.46
GLA P06280 1/20 0.46
RCE1 Q9Y256 1/20 0.46
RAD52 P43351 2/20 0.44
PKM P14618 1/20 0.42
GPR84 Q9NQS5 1/20 0.41
SMPD1 P17405 3/20 0.41
MAPK10 P53779 1/20 0.41
CNR2 P34972 1/20 0.41
ALDH1A1 P00352 2/20 0.41
GAA P10253 1/20 0.41
MAPT P10636 1/20 0.41
MAOA P21397 1/20 0.41
THRA P10827 1/20 0.41
THRB P10828 1/20 0.41
MEN1 O00255 1/20 0.40
MAPK1 P28482 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7991183 0.86 KDM4E (0.49) KDM4EHPGDKMT2AHSD17B10GLA
SCHEMBL7988142 0.85 KDM4E (0.53) KDM4EHPGDKMT2AHSD17B10GLA
SCHEMBL7991327 0.84 KDM4E (0.52) KDM4EHPGDKMT2AHSD17B10GLA
SCHEMBL7991051 0.83 KDM4E (0.50) KDM4EHPGDKMT2AHSD17B10GLA
SCHEMBL7989163 0.82 PTPN11 (0.48) SMPD1THRATHRBMAPK1
SCHEMBL7991229 0.82 KDM4E (0.49) KDM4EHPGDKMT2AHSD17B10GLA
SCHEMBL7991331 0.81 KDM4E (0.53) KDM4EHPGDKMT2AHSD17B10GLA
SCHEMBL7977331 0.80 KDM4E (0.49) KDM4EHPGDKMT2AHSD17B10GLA
SCHEMBL7992415 0.79 KDM4E (0.51) KDM4EHPGDKMT2AHSD17B10GLA
SCHEMBL7987500 0.79 SMPD1 (0.53) KDM4EHPGDKMT2AHSD17B10GLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001055117-A1 NOVEL ISOQUINOLINE DERIVATIVES, PREPARATION METHOD AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM LES LABORATOIRES SERVIER (FR) 2001-08-02 WO disclosed