SCHEMBL7991183

SCHEMBL7991183

C=C(C)CCOc1cc2c(cc1OC)C(C(=O)c1ccccc1)=NCC2

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.49
HPGD P15428 1/20 0.49
KMT2A Q03164 2/20 0.44
HSD17B10 Q99714 2/20 0.44
GLA P06280 1/20 0.44
RCE1 Q9Y256 1/20 0.44
RAD52 P43351 2/20 0.43
ALDH1A1 P00352 3/20 0.40
NR1I2 O75469 2/20 0.40
PKM P14618 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
MAPK10 P53779 2/20 0.40
MAPT P10636 2/20 0.39
GAA P10253 1/20 0.39
MAOA P21397 1/20 0.39
MEN1 O00255 1/20 0.39
MAPK1 P28482 1/20 0.39
LMNA P02545 2/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
CYP1A2 P05177 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7991453 0.86 KDM4E (0.51) KDM4EHPGDKMT2AHSD17B10GLA
SCHEMBL7988142 0.84 KDM4E (0.53) KDM4EHPGDKMT2AHSD17B10GLA
SCHEMBL7991051 0.83 KDM4E (0.50) KDM4EHPGDKMT2AHSD17B10GLA
SCHEMBL7991327 0.83 KDM4E (0.52) KDM4EHPGDKMT2AHSD17B10GLA
SCHEMBL7995609 0.83 S1PR1 (0.40) KDM4EGAAMAOAMAPK1LMNA
SCHEMBL7991229 0.80 KDM4E (0.49) KDM4EHPGDKMT2AHSD17B10GLA
SCHEMBL7991331 0.79 KDM4E (0.53) KDM4EHPGDKMT2AHSD17B10GLA
SCHEMBL7977331 0.78 KDM4E (0.49) KDM4EHPGDKMT2AHSD17B10GLA
SCHEMBL7994703 0.78 KDM4E (0.45) KDM4EHPGDKMT2AHSD17B10GLA
SCHEMBL7992415 0.78 KDM4E (0.51) KDM4EHPGDKMT2AHSD17B10GLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001055117-A1 NOVEL ISOQUINOLINE DERIVATIVES, PREPARATION METHOD AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM LES LABORATOIRES SERVIER (FR) 2001-08-02 WO disclosed