SCHEMBL7991698

SCHEMBL7991698

COc1cc2c(C(=O)c3ccccc3O)nccc2cc1OCc1ccccc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 4/20 0.57
SENP6 Q9GZR1 4/20 0.57
SENP8 Q96LD8 3/20 0.57
SENP7 Q9BQF6 3/20 0.57
APAF1 O14727 2/20 0.57
NSD2 O96028 2/20 0.57
TDP2 O95551 1/20 0.57
PPP1CA P62136 1/20 0.57
SAE1 Q9UBE0 1/20 0.57
UBA2 Q9UBT2 1/20 0.57
L3MBTL1 Q9Y468 1/20 0.54
LMNA P02545 1/20 0.53
SRD5A1 P18405 2/20 0.47
SRD5A2 P31213 2/20 0.47
PDE10A Q9Y233 2/20 0.44
CTSV O60911 2/20 0.44
CTSL P07711 2/20 0.44
PDE3B Q13370 1/20 0.44
PDE3A Q14432 1/20 0.44
KDM4E B2RXH2 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7991450 0.87 CASP3 (0.65) CASP3SENP6SENP8SENP7APAF1
SCHEMBL7991616 0.86 CASP3 (0.64) CASP3SENP6SENP8SENP7APAF1
SCHEMBL7991749 0.84 CASP3 (0.61) CASP3SENP6SENP8SENP7APAF1
SCHEMBL7995165 0.81 CASP3 (0.60) CASP3SENP6SENP8SENP7APAF1
SCHEMBL23457419 0.78 CASP3 (0.66) CASP3SENP6SENP8SENP7APAF1
SCHEMBL23458036 0.78 CASP3 (0.76) CASP3SENP6SENP8SENP7APAF1
SCHEMBL21951885 0.76 MRGPRX1 (0.49) LMNASRD5A1SRD5A2PDE10ACTSV
SCHEMBL27392243 0.75 SRD5A1 (0.53) LMNASRD5A1SRD5A2CTSVCTSL
SCHEMBL1202918 0.73 CASP3 (0.68) CASP3SENP6SENP8SENP7APAF1
SCHEMBL30465578 0.73 KDM1A (0.52) LMNACTSVCTSLKDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001055117-A1 NOVEL ISOQUINOLINE DERIVATIVES, PREPARATION METHOD AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM LES LABORATOIRES SERVIER (FR) 2001-08-02 WO disclosed