SCHEMBL7991781

SCHEMBL7991781

CNCc1cc(C(F)(F)F)cc(C(F)(F)F)c1.CSc1ncc(C(=O)O)c(-c2ccccc2Cl)n1

nearest known ligand 0.47

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
EPAS1 Q99814 1/20 0.43
THRB P10828 3/20 0.43
LMNA P02545 2/20 0.42
TACR1 P25103 5/20 0.42
RXFP1 Q9HBX9 5/20 0.42
POLB P06746 1/20 0.41
JUN P05412 1/20 0.39
NFKB1 P19838 1/20 0.39
NFKB2 Q00653 1/20 0.39
RELA Q04206 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6016692 0.91 TACR1 (0.46) THRBTACR1RXFP1
SCHEMBL6016647 0.90 RXFP1 (0.44) THRBLMNATACR1RXFP1
SCHEMBL6016509 0.90 RXFP1 (0.42) THRBLMNATACR1RXFP1POLB
SCHEMBL6016386 0.89 RXFP1 (0.45) THRBLMNATACR1RXFP1
SCHEMBL7991077 0.88 RXFP1 (0.42) THRBTACR1RXFP1
SCHEMBL6016360 0.85 RXFP1 (0.44) THRBLMNATACR1RXFP1
SCHEMBL6016482 0.83 RXFP1 (0.55) THRBLMNATACR1RXFP1POLB
SCHEMBL6016328 0.81 RXFP1 (0.53) THRBLMNARXFP1POLB
SCHEMBL7991783 0.79 TACR1 (0.49) EPAS1TACR1
SCHEMBL6016462 0.76 CETP (0.43) TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6274588-B1 NEUROKININ OR SUBSTANCE P ANTAGONISTS; CENTRAL NERVOUS SYSTEM AND PSYCHOLOGICAL DISORDES; ANTIDEPRESSANTS, ANXIOLYTIC AGENTS HOFFMANN-LA ROCHE INC. 2001-08-14 US disclosed