SCHEMBL7992280

SCHEMBL7992280

CC(C)(C)OC(=O)N1CCC2(CC1)CN(Cc1cccc(OC(F)(F)F)c1)C(=O)O2

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 4/20 0.42
MGLL Q99685 2/20 0.42
AMPD2 Q01433 1/20 0.42
GPR119 Q8TDV5 3/20 0.41
ENPP2 Q13822 1/20 0.40
TACR1 P25103 1/20 0.40
HCRTR1 O43613 1/20 0.40
HCRTR2 O43614 1/20 0.40
HDAC1 Q13547 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
DRD2 P14416 1/20 0.39
DRD4 P21917 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1086239 0.85 GPR119 (0.43) ROCK2GPR119HDAC1HDAC8HDAC6
SCHEMBL1086688 0.85 OPRD1 (0.50) MGLLGPR119TACR1HDAC1HDAC8
SCHEMBL12184398 0.85 GPR119 (0.45) ROCK2GPR119HDAC1HDAC8HDAC6
SCHEMBL1086247 0.83 GPR119 (0.45) GPR119TACR1HDAC1HDAC8HDAC6
SCHEMBL1086563 0.82 MEN1 (0.47)
SCHEMBL18422018 0.81 MGLL (0.47) MGLLGPR119TACR1HDAC1HDAC8
SCHEMBL7844898 0.80 TACR1 (0.47) ROCK2AMPD2TACR1HCRTR1HCRTR2
SCHEMBL1086929 0.79 MGLL (0.45) MGLLENPP2
SCHEMBL12184200 0.79 HDAC1 (0.52) GPR119HDAC1HDAC8HDAC6
SCHEMBL1086449 0.78 MGLL (0.44) MGLLAMPD2ENPP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6172076-B1 HETEROCYCLE-SUBSTITUTED 1,3,8-TRIAZASPIRO(4,5)DECANE DERIVATIVES; TREATING ARTERIOSCLEROSIS MERCK & CO., INC. 2001-01-09 US disclosed