SCHEMBL7993126

SCHEMBL7993126

O=C1N(CCCCN2CCN(c3csc4ccccc34)CC2)CS(=O)(=O)C12CCCCC2

nearest known ligand 0.68

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 6/20 0.47
HTR1A P08908 5/20 0.47
DRD2 P14416 5/20 0.47
HTR2C P28335 1/20 0.46
ADRA1A P35348 1/20 0.46
HRH1 P35367 1/20 0.46
KCNH2 Q12809 1/20 0.46
DRD4 P21917 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9297541 0.87 HTR2A (0.61) HTR2AHTR1ADRD2ADRA1ADRD4
SCHEMBL7990156 0.80 HTR2A (0.51) HTR2AHTR1ADRD2HTR2CADRA1A
Fumaric Acid SCHEMBL7990225 0.75 HTR2A (0.45) HTR2AHTR1ADRD2HTR2CADRA1A
Maleic Acid SCHEMBL7990218 0.75 HTR2A (0.45) HTR2AHTR1ADRD2HTR2CADRA1A
Maleic Acid SCHEMBL7993166 0.74 HTR2A (0.46) HTR2AHTR1ADRD2HTR2CADRA1A
Fumaric Acid SCHEMBL7993170 0.74 HTR2A (0.46) HTR2AHTR1ADRD2HTR2CADRA1A
SCHEMBL7993408 0.74 HTR2A (0.65) HTR2AHTR1ADRD2ADRA1ADRD4
SCHEMBL9380372 0.72 HTR1A (0.50) HTR2AHTR1ADRD2ADRA1AHRH1
SCHEMBL9381448 0.72 HTR1A (0.76) HTR2AHTR1ADRD2ADRA1ADRD4
Hydrochloric Acid SCHEMBL9380816 0.71 HTR1A (0.74) HTR2AHTR1ADRD2DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6284775-B1 PSYCHOLOGICAL DISORDERS AVENTIS PHARMACEUTICALS INC. 2001-09-04 US disclosed
US-5371087-A Antipsychotic, analgesics, anticonvulsant and anxiolytic agent HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1994-12-06 US disclosed
US-5229388-A 3-[4-(1-substituted-4-piperazinyl)butyl]-4-thiazolidinone and related compounds HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1993-07-20 US disclosed