SCHEMBL7993392

SCHEMBL7993392

Fc1ccc2cc(C3CNCCN3)sc2c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 4/20 0.36
HTR2A P28223 2/20 0.36
SLC6A4 P31645 2/20 0.35
SLC6A2 P23975 1/20 0.35
SLC6A3 Q01959 1/20 0.35
KCNH2 Q12809 1/20 0.35
ROCK2 O75116 1/20 0.33
ROCK1 Q13464 1/20 0.33
HTR2B P41595 2/20 0.33
MPO P05164 1/20 0.32
HTR1A P08908 2/20 0.31
BRAF P15056 1/20 0.31
CHRNA7 P36544 2/20 0.31
HTR3A P46098 2/20 0.31
AXL P30530 1/20 0.31
GFER P55789 1/20 0.31
CHRNB2 P17787 1/20 0.31
CHRNB4 P30926 1/20 0.31
CHRNA3 P32297 1/20 0.31
CHRNA4 P43681 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7997135 0.84 HTR2C (0.37) HTR2CHTR2ASLC6A4SLC6A2KCNH2
Hydrochloric Acid SCHEMBL2957747 0.82 HTR2C (0.36) HTR2CHTR2AKCNH2HTR2BHTR1A
SCHEMBL7993434 0.82 HTR2A (0.40) HTR2CHTR2ASLC6A4SLC6A2SLC6A3
Hydrochloric Acid SCHEMBL8688971 0.81 HTR2A (0.42) HTR2CHTR2ASLC6A4SLC6A2SLC6A3
SCHEMBL5760443 0.75 SLC6A4 (0.40) SLC6A4SLC6A2SLC6A3KCNH2MPO
SCHEMBL16644685 0.74 ROCK2 (0.34) ROCK2ROCK1
Hydrochloric Acid SCHEMBL7108504 0.74 NPC1 (0.40) HTR2CHTR2ASLC6A4SLC6A2SLC6A3
SCHEMBL7993389 0.72 MAPT (0.36) HTR2CHTR2AKCNH2CHRNB2CHRNB4
SCHEMBL4536065 0.70 CHRNB2 (0.42) HTR2CHTR2ASLC6A4SLC6A2SLC6A3
SCHEMBL27608178 0.70 BACE1 (0.41) HTR2CHTR2ASLC6A4SLC6A2SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6284775-B1 PSYCHOLOGICAL DISORDERS AVENTIS PHARMACEUTICALS INC. 2001-09-04 US disclosed
EP-0511610-B1 Benzisothiazole- and benzisoxazole-3-carboxamides, a process for their preparation and their use as antipsychotic medicaments HOECHST ROUSSEL PHARMA (US) 1996-09-11 EP disclosed
US-5371087-A Antipsychotic, analgesics, anticonvulsant and anxiolytic agent HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1994-12-06 US disclosed
US-5229388-A 3-[4-(1-substituted-4-piperazinyl)butyl]-4-thiazolidinone and related compounds HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1993-07-20 US disclosed
EP-0511610-A1 Benzisothiazole- and benzisoxazole-3-carboxamides, a process for their preparation and their use as antipsychotic medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1992-11-04 EP disclosed
US-5143923-A Psychological disorders HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1992-09-01 US disclosed
US-5136037-A 3-(4-substituted-4-piperazinyl)butyl-4-thiazolidinone and related compounds HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1992-08-04 US disclosed
US-5037984-A Anticonvulsants; anxiolytic agents HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1991-08-06 US disclosed
US-4933453-A ANTIPSYCHOTIC, ANALGESIC, ANTICONVULSANT, AND ANXIOLYTIC AGENTS HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1990-06-12 US disclosed