SCHEMBL7993416

SCHEMBL7993416

CC1N(CCCCN2CCN(c3ncccn3)CC2)C(=O)CS1(=O)=O

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 6/20 0.54
DRD2 P14416 4/20 0.54
HTR2A P28223 3/20 0.54
ABCB11 O95342 2/20 0.49
ALDH1A1 P00352 2/20 0.49
CYP1A2 P05177 2/20 0.49
CYP2D6 P10635 2/20 0.49
ADRA2C P18825 2/20 0.49
DRD4 P21917 2/20 0.49
ADRA1D P25100 2/20 0.49
HTR7 P34969 2/20 0.49
ADRA1A P35348 2/20 0.49
ADRA1B P35368 2/20 0.49
DRD3 P35462 2/20 0.49
ADRA2A P08913 1/20 0.49
ADRA2B P18089 1/20 0.49
CYP2C19 P33261 1/20 0.49
HTR6 P50406 1/20 0.49
SLC22A2 O15244 1/20 0.49
CYP3A4 P08684 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7989840 0.77 HTR1A (0.55) HTR1ADRD2HTR2AABCB11ALDH1A1
SCHEMBL26492991 0.74 HTR1A (0.65) HTR1ADRD2HTR2AABCB11ALDH1A1
SCHEMBL26108581 0.74 HTR1A (0.65) HTR1ADRD2HTR2AABCB11ALDH1A1
SCHEMBL10753571 0.74 HTR1A (0.54) HTR1ADRD2HTR2AABCB11ALDH1A1
Hydrochloric Acid SCHEMBL26108377 0.73 DRD2 (0.63) HTR1ADRD2HTR2AALDH1A1DRD3
SCHEMBL9197820 0.71 DRD2 (0.61) HTR1ADRD2HTR2ADRD4
SCHEMBL10784615 0.71 DRD2 (0.70) HTR1ADRD2HTR2ADRD4
SCHEMBL9589567 0.71 DRD2 (0.67) HTR1ADRD2DRD4
SCHEMBL10784007 0.71 DRD2 (0.67) HTR1ADRD2DRD4
SCHEMBL10788382 0.71 DRD2 (0.74) HTR1ADRD2HTR2ADRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6284775-B1 PSYCHOLOGICAL DISORDERS AVENTIS PHARMACEUTICALS INC. 2001-09-04 US disclosed
US-5371087-A Antipsychotic, analgesics, anticonvulsant and anxiolytic agent HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1994-12-06 US disclosed
US-5229388-A 3-[4-(1-substituted-4-piperazinyl)butyl]-4-thiazolidinone and related compounds HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1993-07-20 US disclosed